PRACTICAL TOTAL SYNTHESIS OF RS-15385

被引：23

作者：

ROHLOFF, JC

DYSON, NH

GARDNER, JO

ALFREDSON, TV

SPARACINO, ML

ROBINSON, J

机构：

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1993年 / 58卷 / 07期

关键词：

D O I：

10.1021/jo00059a056

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

收藏

页码：1935 / 1938

页数：4

相关论文

共 18 条

[1]

AKHREM AA, 1980, SYNTHESIS-STUTTGART, P996

[2]

BROWN CM, 1990, BRIT J PHARMACOL, V99, pP272

[3] SELECTIVE REDUCTIONS .18. FAST REACTION OF PRIMARY, SECONDARY, AND TERTIARY AMIDES WITH DIBORANE - SIMPLE, CONVENIENT PROCEDURE FOR CONVERSION OF AMIDES TO CORRESPONDING AMINES [J].

BROWN, HC ;

HEIM, P .

JOURNAL OF ORGANIC CHEMISTRY, 1973, 38 (05) :912-916

[4]

Clark R D, 1986, Prog Med Chem, V23, P1, DOI 10.1016/S0079-6468(08)70339-4

[5] (8A-ALPHA,12A-ALPHA,13A-ALPHA)-5,8,8A,9,10,11,12,12A,13,13A-DECAHYDRO-3-METHOXY-12-(METHYLSULFONYL)-6H-ISOQUINO[2,1-G][1,6]NAPHTHYRIDINE, A POTENT AND HIGHLY SELECTIVE ALPHA2-ADRENOCEPTOR ANTAGONIST [J].

CLARK, RD ;

REPKE, DB ;

KILPATRICK, AT ;

BROWN, CM ;

MACKINNON, AC ;

CLAGUE, RU ;

SPEDDING, M .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (09) :2034-2036

[6]

CLARK RD, 1990, HETEROCYCLES, V31, P353

[7] STRUCTURE AFFINITY RELATIONSHIPS OF 12-SULFONYL DERIVATIVES OF 5,8,8A,9,10,11,12,12A,13,13A-DECAHYDRO-6H-ISOQUINO[2,1-G][1,6]NAPHTHYRIDINES AT ALPHA-ADRENOCEPTORS [J].

CLARK, RD ;

REPKE, DB ;

BERGER, J ;

NELSON, JT ;

KILPATRICK, AT ;

BROWN, CM ;

MACKINNON, AC ;

CLAGUE, RU ;

SPEDDING, M .

JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (02) :705-717

[8]

CLARK RD, 1990, BRIT J PHARMACOL, V99, pP123

[9] FLUORESZENZMETHODEN ZUR HISTOCHEMISCHEN SICHTBARMACHUNG VON MONOAMINEN .6. IDENTIFIZIERUNG DER FLUORESZIERENDEN PRODUKTE AUS M-HYDROXY-PHENYLATHYLAMINEN UND FORMALDEHYD [J].

CORRODI, H ;

JONSSON, G .

HELVETICA CHIMICA ACTA, 1966, 49 (01) :798-+

[10] ENANTIOMERIC PURITY DETERMINATION OF 3-AMINOQUINUCLIDINE BY DIASTEREOMERIC DERIVATIZATION AND HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC SEPARATION [J].

DEMIAN, I ;

GRIPSHOVER, DF .

JOURNAL OF CHROMATOGRAPHY, 1989, 466 :415-420