INFLUENCE OF SUBSTRATE CONCENTRATION ON THE PHASE-I AND PHASE-II METABOLISM OF 4-METHOXYBIPHENYL BY RAT ISOLATED HEPATOCYTES

被引:2
作者
FRY, JR
机构
关键词
D O I
10.3109/00498258709043982
中图分类号
R9 [药学];
学科分类号
1007 ;
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页码:751 / 758
页数:8
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共 15 条
[1]  
CAMPBELL RC, 1967, STATISTICS BIOL, P49
[2]   BIOTRANSFORMATION OF 4-DIMETHYLAMINOPHENOL IN ISOLATED PERFUSED RAT-LIVER AND IN RAT [J].
EYER, P ;
KAMPFFMEYER, HG .
BIOCHEMICAL PHARMACOLOGY, 1978, 27 (18) :2223-2228
[3]  
Fry J R, 1981, Methods Enzymol, V77, P130
[4]  
FRY JR, 1981, BIOCHEM PHARMACOL, V30, P1915, DOI 10.1016/0006-2952(81)90199-4
[5]   SULFOCONJUGATION AND GLUCURONIDATION OF SALICYLAMIDE IN ISOLATED RAT HEPATOCYTES [J].
KOIKE, M ;
SUGENO, K ;
HIRATA, M .
JOURNAL OF PHARMACEUTICAL SCIENCES, 1981, 70 (03) :308-311
[6]   KINETICS OF SULFATION AND GLUCURONIDATION OF HARMOL IN THE PERFUSED-RAT-LIVER PREPARATION - DISAPPEARANCE OF ABERRANCES IN GLUCURONIDATION KINETICS BY INHIBITION OF SULFATION [J].
KOSTER, H ;
HALSEMA, I ;
SCHOLTENS, E ;
PANG, KS ;
MULDER, GJ .
BIOCHEMICAL PHARMACOLOGY, 1982, 31 (19) :3023-3028
[7]  
KOSTER H, 1982, DRUG METAB DISPOS, V10, P330
[8]   DOSE-DEPENDENT SHIFTS IN THE SULFATION AND GLUCURONIDATION OF PHENOLIC-COMPOUNDS IN THE RAT INVIVO AND IN ISOLATED HEPATOCYTES - THE ROLE OF SATURATION OF PHENOLSULFOTRANSFERASE [J].
KOSTER, H ;
HALSEMA, I ;
SCHOLTENS, E ;
KNIPPERS, M ;
MULDER, GJ .
BIOCHEMICAL PHARMACOLOGY, 1981, 30 (18) :2569-2575
[9]  
LEVY G, 1967, J PHARMACOL EXP THER, V156, P285
[10]   INTERRELATIONSHIP BETWEEN DEMETHYLATION OF P-NITROANISOLE AND CONJUGATION OF P-NITROPHENOL IN RAT-LIVER [J].
MINCK, K ;
SCHUPP, RR ;
ILLING, HPA ;
KAHL, GF ;
NETTER, KJ .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1973, 279 (04) :347-360