SPECIFICITY OF ESTERASES AND STRUCTURE OF PRODRUG ESTERS - REACTIVITY OF VARIOUS ACYLATED ACETAMINOPHEN COMPOUNDS AND ACETYLAMINOBENZOATED COMPOUNDS

被引：18

作者：

SEKI, H

KAWAGUCHI, T

HIGUCHI, T

机构：

[1] TEIJIN LTD,INST BIOMED RES,HINO,TOKYO 191,JAPAN

[2] UNIV KANSAS,DEPT PHARMACEUT CHEM,LAWRENCE,KS 66045

来源：

JOURNAL OF PHARMACEUTICAL SCIENCES | 1988年 / 77卷 / 10期

关键词：

D O I：

10.1002/jps.2600771009

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：855 / 860

页数：6

共 10 条

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[3]

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[4]

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[5]

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[6]

McLafferty F. W., 1973, IMTERPRETATION MASS, P156

[7] 4-DIALKYLAMINOPYRIDINES AS ACYLATION CATALYSTS .5. SIMPLE METHOD FOR ESTERIFICATION OF CARBOXYLIC-ACIDS [J].

NEISES, B ;

STEGLICH, W .

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 1978, 17 (07) :522-524

[8] RATIONALE FOR DESIGN OF BIOLOGICALLY REVERSIBLE DRUG DERIVATIVES - PRODRUGS [J].

SINKULA, AA ;

YALKOWSKY, SH .

JOURNAL OF PHARMACEUTICAL SCIENCES, 1975, 64 (02) :181-210

[9]

STELLA VJ, 1985, DIRECTED DRUG DELIVE, P247

[10]

WOODS RJ, UNPUB

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