A RAPID ENTRY INTO PODOPHYLLOTOXIN CONGENERS - SYNTHESIS OF JUSTICIDIN-B

被引：15

作者：

KAMAL, A ^{[1
]}

DANESHTALAB, M ^{[1
]}

MICETICH, RG ^{[1
]}

机构：

[1] SYNPHAR LABS INC, EDMONTON T6E 5V2, AB, CANADA

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 23期

关键词：

PODOPHYLLOTOXIN; PODOPHYLLUM LIGNANS; JUSTICIDIN B; MICHAEL INITIATED RING CLOSURE; DESULFURIZATION; NICKEL-CONTAINING; COMPLEX REDUCING AGENT;

D O I：

10.1016/S0040-4039(00)76691-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A facile synthesis of justicidin B is described, as well as related podophyllum lignans by employing Michael Initiated Ring Closure strategy followed by desulfurization mediated by nickel-containing complex reducing agent.

引用

页码：3879 / 3882

页数：4

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