REGIOSELECTIVE IMIDE REDUCTION - AN ISSUE IN THE TOTAL SYNTHESIS OF STAUROSPORINE

被引：34

作者：

LINK, JT

DANISHEFSKY, SJ

机构：

[1] COLUMBIA UNIV,DEPT CHEM,NEW YORK,NY 10027

[2] MEM SLOAN KETTERING CANC CTR,SLOAN KETTERING INST CANC RES,BIOORGAN CHEM LAB,NEW YORK,NY 10021

来源：

TETRAHEDRON LETTERS | 1994年 / 35卷 / 49期

关键词：

D O I：

10.1016/0040-4039(94)88446-3

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An imide was regioselectively reduced to either of its corresponding lactams. These lactams serve as potent glycosyl accepters and can be converted into the aglycone of staurosporine.

引用

页码：9135 / 9138

页数：4

共 12 条

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