GABA(B) RECEPTOR ANTAGONISTS - FROM SYNTHESIS TO THERAPEUTIC APPLICATIONS

被引:107
作者
BITTIGER, H
FROESTL, W
MICKEL, SJ
OLPE, HR
机构
[1] Research and Development, Pharmaceuticals Division, Ciba-Geigy Ltd.
关键词
D O I
10.1016/0165-6147(93)90056-P
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:391 / 394
页数:4
相关论文
共 25 条
  • [21] CGP 35348 - A CENTRALLY ACTIVE BLOCKER OF GABA-B RECEPTORS
    OLPE, HR
    KARLSSON, G
    POZZA, MF
    BRUGGER, F
    STEINMANN, M
    VANRIEZEN, H
    FAGG, G
    HALL, RG
    FROESTL, W
    BITTIGER, H
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1990, 187 (01) : 27 - 38
  • [22] THE ACTIONS OF ORALLY ACTIVE GABA(B) RECEPTOR ANTAGONISTS ON GABAERGIC TRANSMISSION INVIVO AND INVITRO
    OLPE, HR
    STEINMANN, MW
    FERRAT, T
    POZZA, MF
    GREINER, K
    BRUGGER, F
    FROESTL, W
    MICKEL, SJ
    BITTIGER, H
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1993, 233 (2-3) : 179 - 186
  • [23] REPEATED ADMINISTRATION OF DESIPRAMINE AND A GABA(B) RECEPTOR ANTAGONIST, CGP-36742, DISCRETELY UP-REGULATES GABA(B) RECEPTOR-BINDING SITES IN RAT FRONTAL-CORTEX
    PRATT, GD
    BOWERY, NG
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1993, 110 (02) : 724 - 735
  • [24] WALDMEIER PC, 1990, GABAB RECEPTORS IN MAMMALIAN FUNCTION, P63
  • [25] WALDMEIER PC, 1992, PHARM COMMUN, V2, P4