PHYSICOCHEMICAL PROPERTY MODIFICATION STRATEGIES BASED ON ENZYME SUBSTRATE SPECIFICITIES .1. RATIONALE, SYNTHESIS, AND PHARMACEUTICAL PROPERTIES OF ASPIRIN DERIVATIVES

被引：23

作者：

BANERJEE, PK ^{[1
]}

AMIDON, GL ^{[1
]}

机构：

[1] UNIV WISCONSIN,SCH PHARM,MADISON,WI 53706

来源：

JOURNAL OF PHARMACEUTICAL SCIENCES | 1981年 / 70卷 / 12期

关键词：

D O I：

10.1002/jps.2600701202

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：1299 / 1303

页数：5

共 19 条

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AMIDON, GL .

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[5] PHYSICOCHEMICAL PROPERTY MODIFICATION STRATEGIES BASED ON ENZYME SUBSTRATE SPECIFICITIES .3. CARBOXYPEPTIDASE A-HYDROLYSIS OF ASPIRIN DERIVATIVES [J].

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AMIDON, GL .

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[6] BLOOD CONCENTRATION PROFILES OF ACETAMINOPHEN FOLLOWING ORAL-ADMINISTRATION OF FATTY-ACID ESTERS OF ACETAMINOPHEN WITH PANCREATIC LIPASE TO DOGS [J].

BAUGUESS, CT ;

FINCHER, JH ;

SADIK, F ;

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[7]

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[8]

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[9]

DAVISON C, 1966, CLIN PHARM THER, V7, P329

[10] THE HYDROLYSIS OF ASPIRIN - A DETERMINATION OF THE THERMODYNAMIC DISSOCIATION CONSTANT AND A STUDY OF THE REACTION KINETICS BY ULTRA-VIOLET SPECTROPHOTOMETRY [J].

EDWARDS, LJ .

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