IRREVERSIBLE ENZYME INHIBITORS .90. CANDIDATE ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITORS OF THYMIDYLATE SYNTHETASE .I. 2-AMINO-5-(BENZENESULFONAMIDOPROPYL)-6-METHYL-4-PYRIMIDINOL WITH SUBSTITUENTS ON BENZENE RING (1,2)

被引：4

作者：

BAKER, BR

COWARD, JK

机构：

来源：

JOURNAL OF HETEROCYCLIC CHEMISTRY | 1967年 / 4卷 / 02期

关键词：

D O I：

10.1002/jhet.5570040206

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：195 / &

共 32 条

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[6] ANALOGS OF TETRAHYDROFOLIC ACID .20. EFFECTS OF MODIFICATION OF BRIDGE BETWEEN PYRIMIDYL AND PHENYL MOIETIES OF 2-AMINO-5-(3-ANILINOPROPYL)-6-METHYL-4-PYRIMIDINOL ON INHIBITION OF DIHYDROFOLIC REDUCTASE AND THYMIDYLATE SYNTHETASE 2 [J].

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[7] IRREVERSIBLE ENZYME INHIBITORS .89. CANDIDATE ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITORS OF DIHYDROFOLIC REDUCTASE .X. DERIVATIVES OF 2-AMINO-5-BENZAMIDOPROPYL-4-PYRIMIDINOL (1,2) [J].

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[9] IRREVERSIBLE ENZYME INHIBITORS .68. 2-AMINO-5-(P-BROMOACETAMIDOPHENOXYPROPYL)-6-PHENYL-4-PYRIMIDINOL AN ACTIVE-SITE-DIRECTED IRREVERSIBLE INHIBITOR OF DIHYDROFOLIC REDUCTASE [J].

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[10]

BAKER BR, 1966, J PHARM SCI, V55, P1417, DOI 10.1002/jps.2600551218

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