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CGS-24128 - A LONG-ACTING INHIBITOR OF NEUTRAL ENDOPEPTIDASE-3.4.24.11
被引:6
作者
:
TRAPANI, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
Research Department, Pharmaceuticals Division, CIBA-GEIGY Corporation, Summit, New Jersey
TRAPANI, AJ
SMITS, JFM
论文数:
0
引用数:
0
h-index:
0
机构:
Research Department, Pharmaceuticals Division, CIBA-GEIGY Corporation, Summit, New Jersey
SMITS, JFM
SUN, XJ
论文数:
0
引用数:
0
h-index:
0
机构:
Research Department, Pharmaceuticals Division, CIBA-GEIGY Corporation, Summit, New Jersey
SUN, XJ
WEBB, RL
论文数:
0
引用数:
0
h-index:
0
机构:
Research Department, Pharmaceuticals Division, CIBA-GEIGY Corporation, Summit, New Jersey
WEBB, RL
YAU, ET
论文数:
0
引用数:
0
h-index:
0
机构:
Research Department, Pharmaceuticals Division, CIBA-GEIGY Corporation, Summit, New Jersey
YAU, ET
机构
:
[1]
Research Department, Pharmaceuticals Division, CIBA-GEIGY Corporation, Summit, New Jersey
来源
:
CARDIOVASCULAR DRUG REVIEWS
|
1994年
/ 12卷
/ 04期
关键词
:
ANGIOTENSIN-CONVERTING ENZYME;
ATRIAL NATRIURETIC PEPTIDE;
CGS;
24128;
25462;
ENZYME INHIBITORS;
HEART FAILURE;
HYPERTENSION;
NEUTRAL ENDOPEPTIDASE 3.4.24.11;
D O I
:
10.1111/j.1527-3466.1994.tb00294.x
中图分类号
:
R5 [内科学];
学科分类号
:
1002 ;
100201 ;
摘要
:
[No abstract available]
引用
收藏
页码:271 / 285
页数:15
相关论文
共 58 条
[51]
THIORPHAN, AN INHIBITOR OF ENDOPEPTIDASE 24.11, POTENTIATES THE NATRIURETIC ACTIVITY OF ATRIAL NATRIURETIC PEPTIDE
[J].
TRAPANI, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
TRAPANI, AJ
;
SMITS, GJ
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
SMITS, GJ
;
MCGRAW, DE
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
MCGRAW, DE
;
SPEAR, KL
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
SPEAR, KL
;
KOEPKE, JP
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
KOEPKE, JP
;
OLINS, GM
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
OLINS, GM
;
BLAINE, EH
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
BLAINE, EH
.
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1989,
14
(03)
:419
-424
[52]
PHARMACOLOGICAL PROFILE OF CGS-24128, A POTENT, LONG-ACTING INHIBITOR OF NEUTRAL ENDOPEPTIDASE-24.11
[J].
TRAPANI, AJ
论文数:
0
引用数:
0
h-index:
0
TRAPANI, AJ
;
BELL, ME
论文数:
0
引用数:
0
h-index:
0
BELL, ME
;
COTE, DT
论文数:
0
引用数:
0
h-index:
0
COTE, DT
;
DELOMBAERT, S
论文数:
0
引用数:
0
h-index:
0
DELOMBAERT, S
;
ERION, MD
论文数:
0
引用数:
0
h-index:
0
ERION, MD
;
GERLOCK, TE
论文数:
0
引用数:
0
h-index:
0
GERLOCK, TE
;
GHAI, RD
论文数:
0
引用数:
0
h-index:
0
GHAI, RD
;
HOPKINS, MF
论文数:
0
引用数:
0
h-index:
0
HOPKINS, MF
;
PEPPARD, JV
论文数:
0
引用数:
0
h-index:
0
PEPPARD, JV
;
WEBB, RL
论文数:
0
引用数:
0
h-index:
0
WEBB, RL
;
LAPPE, RW
论文数:
0
引用数:
0
h-index:
0
LAPPE, RW
;
WORCEL, M
论文数:
0
引用数:
0
h-index:
0
WORCEL, M
.
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1994,
23
(03)
:358
-364
[53]
TRAPANI AJ, 1993, BIOCHEM MOL BIOL INT, V31, P861
[54]
ANTIHYPERTENSIVE ACTION OF THE CONVERTING-ENZYME-INHIBITOR PERINDOPRIL (S9490-3) IN SPONTANEOUSLY HYPERTENSIVE RATS - COMPARISON WITH ENALAPRIL (MK421) AND RAMIPRIL (HOE498)
[J].
UNGER, T
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNGER, T
;
MOURSI, M
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
MOURSI, M
;
GANTEN, D
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
GANTEN, D
;
HERMANN, K
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
HERMANN, K
;
LANG, RE
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
LANG, RE
.
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1986,
8
(02)
:276
-285
[55]
DNA-SYNTHESIS IN THE NONINFARCTED CARDIAC INTERSTITIUM AFTER LEFT CORONARY-ARTERY LIGATION IN THE RAT - EFFECTS OF CAPTOPRIL
[J].
VANKRIMPEN, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
VANKRIMPEN, C
;
SMITS, JFM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
SMITS, JFM
;
CLEUTJENS, JPM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
CLEUTJENS, JPM
;
DEBETS, JJM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
DEBETS, JJM
;
SCHOEMAKER, RG
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
SCHOEMAKER, RG
;
BOUDIER, HAJS
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
BOUDIER, HAJS
;
BOSMAN, FT
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
BOSMAN, FT
;
DAEMEN, MJAP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
DAEMEN, MJAP
.
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY,
1991,
23
(11)
:1245
-1253
[56]
DEGRADATION OF ATRIAL NATRIURETIC PEPTIDE - PHARMACOLOGIC EFFECTS OF PROTEASE EC 24.11 INHIBITION
[J].
WEBB, RL
论文数:
0
引用数:
0
h-index:
0
WEBB, RL
;
YASAY, GD
论文数:
0
引用数:
0
h-index:
0
YASAY, GD
;
MCMARTIN, C
论文数:
0
引用数:
0
h-index:
0
MCMARTIN, C
;
MCNEAL, RB
论文数:
0
引用数:
0
h-index:
0
MCNEAL, RB
;
ZIMMERMAN, MB
论文数:
0
引用数:
0
h-index:
0
ZIMMERMAN, MB
.
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1989,
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PATHOLOGICAL HYPERTROPHY AND CARDIAC INTERSTITIUM - FIBROSIS AND RENIN-ANGIOTENSIN-ALDOSTERONE SYSTEM
[J].
WEBER, KT
论文数:
0
引用数:
0
h-index:
0
机构:
Univ. of Missouri-Columbia, Columbia, MO 65212, Medical Sciences Building
WEBER, KT
;
BRILLA, CG
论文数:
0
引用数:
0
h-index:
0
机构:
Univ. of Missouri-Columbia, Columbia, MO 65212, Medical Sciences Building
BRILLA, CG
.
CIRCULATION,
1991,
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MAXIMIZING THE NATRIURETIC EFFECT OF ENDOGENOUS ATRIOPEPTIN IN A RAT MODEL OF HEART-FAILURE
[J].
WILKINS, MR
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,660 S EUCLID,ST LOUIS,MO 63110
WILKINS, MR
;
SETTLE, SL
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,660 S EUCLID,ST LOUIS,MO 63110
SETTLE, SL
;
STOCKMANN, PT
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,660 S EUCLID,ST LOUIS,MO 63110
STOCKMANN, PT
;
NEEDLEMAN, P
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,660 S EUCLID,ST LOUIS,MO 63110
NEEDLEMAN, P
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
1990,
87
(16)
:6465
-6469
←
1
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共 58 条
[51]
THIORPHAN, AN INHIBITOR OF ENDOPEPTIDASE 24.11, POTENTIATES THE NATRIURETIC ACTIVITY OF ATRIAL NATRIURETIC PEPTIDE
[J].
TRAPANI, AJ
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
TRAPANI, AJ
;
SMITS, GJ
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
SMITS, GJ
;
MCGRAW, DE
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
MCGRAW, DE
;
SPEAR, KL
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
SPEAR, KL
;
KOEPKE, JP
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
KOEPKE, JP
;
OLINS, GM
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
OLINS, GM
;
BLAINE, EH
论文数:
0
引用数:
0
h-index:
0
机构:
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
WASHINGTON UNIV,SCH MED,DEPT PHARMACOL,SEARLE RES & DEV,ST LOUIS,MO 63110
BLAINE, EH
.
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1989,
14
(03)
:419
-424
[52]
PHARMACOLOGICAL PROFILE OF CGS-24128, A POTENT, LONG-ACTING INHIBITOR OF NEUTRAL ENDOPEPTIDASE-24.11
[J].
TRAPANI, AJ
论文数:
0
引用数:
0
h-index:
0
TRAPANI, AJ
;
BELL, ME
论文数:
0
引用数:
0
h-index:
0
BELL, ME
;
COTE, DT
论文数:
0
引用数:
0
h-index:
0
COTE, DT
;
DELOMBAERT, S
论文数:
0
引用数:
0
h-index:
0
DELOMBAERT, S
;
ERION, MD
论文数:
0
引用数:
0
h-index:
0
ERION, MD
;
GERLOCK, TE
论文数:
0
引用数:
0
h-index:
0
GERLOCK, TE
;
GHAI, RD
论文数:
0
引用数:
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GHAI, RD
;
HOPKINS, MF
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HOPKINS, MF
;
PEPPARD, JV
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PEPPARD, JV
;
WEBB, RL
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WEBB, RL
;
LAPPE, RW
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LAPPE, RW
;
WORCEL, M
论文数:
0
引用数:
0
h-index:
0
WORCEL, M
.
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1994,
23
(03)
:358
-364
[53]
TRAPANI AJ, 1993, BIOCHEM MOL BIOL INT, V31, P861
[54]
ANTIHYPERTENSIVE ACTION OF THE CONVERTING-ENZYME-INHIBITOR PERINDOPRIL (S9490-3) IN SPONTANEOUSLY HYPERTENSIVE RATS - COMPARISON WITH ENALAPRIL (MK421) AND RAMIPRIL (HOE498)
[J].
UNGER, T
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNGER, T
;
MOURSI, M
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
MOURSI, M
;
GANTEN, D
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
GANTEN, D
;
HERMANN, K
论文数:
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引用数:
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h-index:
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机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
HERMANN, K
;
LANG, RE
论文数:
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引用数:
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h-index:
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机构:
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
UNIV HEIDELBERG,DEPT PHARMACOL,D-6900 HEIDELBERG,FED REP GER
LANG, RE
.
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY,
1986,
8
(02)
:276
-285
[55]
DNA-SYNTHESIS IN THE NONINFARCTED CARDIAC INTERSTITIUM AFTER LEFT CORONARY-ARTERY LIGATION IN THE RAT - EFFECTS OF CAPTOPRIL
[J].
VANKRIMPEN, C
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
VANKRIMPEN, C
;
SMITS, JFM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
SMITS, JFM
;
CLEUTJENS, JPM
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
CLEUTJENS, JPM
;
DEBETS, JJM
论文数:
0
引用数:
0
h-index:
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机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
DEBETS, JJM
;
SCHOEMAKER, RG
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
SCHOEMAKER, RG
;
BOUDIER, HAJS
论文数:
0
引用数:
0
h-index:
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机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
BOUDIER, HAJS
;
BOSMAN, FT
论文数:
0
引用数:
0
h-index:
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机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
BOSMAN, FT
;
DAEMEN, MJAP
论文数:
0
引用数:
0
h-index:
0
机构:
UNIV LIMBURG, DEPT PATHOL, POB 616, 6200 MD MAASTRICHT, NETHERLANDS
DAEMEN, MJAP
.
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY,
1991,
23
(11)
:1245
-1253
[56]
DEGRADATION OF ATRIAL NATRIURETIC PEPTIDE - PHARMACOLOGIC EFFECTS OF PROTEASE EC 24.11 INHIBITION
[J].
WEBB, RL
论文数:
0
引用数:
0
h-index:
0
WEBB, RL
;
YASAY, GD
论文数:
0
引用数:
0
h-index:
0
YASAY, GD
;
MCMARTIN, C
论文数:
0
引用数:
0
h-index:
0
MCMARTIN, C
;
MCNEAL, RB
论文数:
0
引用数:
0
h-index:
0
MCNEAL, RB
;
ZIMMERMAN, MB
论文数:
0
引用数:
0
h-index:
0
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