AN IMPROVED SYNTHETIC ROUTE TO HUPERZINE-A - NEW ANALOGS AND THEIR INHIBITION OF ACETYLCHOLINESTERASE

被引：35

作者：

KOZIKOWSKI, AP ^{[1
]}

CAMPIANI, G ^{[1
]}

AAGAARD, P ^{[1
]}

MCKINNEY, M ^{[1
]}

机构：

[1] MAYO FDN MED EDUC & RES,NEUROPHARMACOL RES,JACKSONVILLE,FL 32224

来源：

JOURNAL OF THE CHEMICAL SOCIETY-CHEMICAL COMMUNICATIONS | 1993年 / 10期

关键词：

D O I：

10.1039/c39930000860

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A bicycloannulation approach to huperzine A is detailed together with syntheses of the methylene analogue 8, the diamino compound 12 and their inhibition of acetylcholinesterase.

引用

页码：860 / 862

页数：3

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