HIV-1-SPECIFIC RT INHIBITORS - HIGHLY SELECTIVE INHIBITORS OF HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1 THAT ARE SPECIFICALLY TARGETED AT THE VIRAL REVERSE-TRANSCRIPTASE

被引:183
作者
DECLERCQ, E
机构
[1] Rega Institute for Medical Research, Katholieke Universiteit Leuven, Leuven
关键词
D O I
10.1002/med.2610130303
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:229 / 258
页数:30
相关论文
共 53 条
  • [31] INHIBITION OF HIV-1 REPLICATION BY A NONNUCLEOSIDE REVERSE-TRANSCRIPTASE INHIBITOR
    MERLUZZI, VJ
    HARGRAVE, KD
    LABADIA, M
    GROZINGER, K
    SKOOG, M
    WU, JC
    SHIH, CK
    ECKNER, K
    HATTOX, S
    ADAMS, J
    ROSEHTHAL, AS
    FAANES, R
    ECKNER, RJ
    KOUP, RA
    SULLIVAN, JL
    [J]. SCIENCE, 1990, 250 (4986) : 1411 - 1413
  • [32] A NOVEL LEAD FOR SPECIFIC ANTI-HIV-1 AGENTS - 1-[(2-HYDROXYETHOXY)METHYL]-6-(PHENYLTHIO)THYMINE
    MIYASAKA, T
    TANAKA, H
    BABA, M
    HAYAKAWA, H
    WALKER, RT
    BALZARINI, J
    DECLERCQ, E
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (12) : 2507 - 2509
  • [33] CRYSTAL-STRUCTURE OF NEVIRAPINE, A NONNUCLEOSIDE INHIBITOR OF HIV-1 REVERSE-TRANSCRIPTASE, AND COMPUTATIONAL ALIGNMENT WITH A STRUCTURALLY DIVERSE INHIBITOR
    MUI, PW
    JACOBER, SP
    HARGRAVE, KD
    ADAMS, J
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (01) : 201 - 202
  • [34] VIRAL RESISTANCE TO HUMAN-IMMUNODEFICIENCY-VIRUS TYPE-1-SPECIFIC PYRIDINONE REVERSE-TRANSCRIPTASE INHIBITORS
    NUNBERG, JH
    SCHLEIF, WA
    BOOTS, EJ
    OBRIEN, JA
    QUINTERO, JC
    HOFFMAN, JM
    EMINI, EA
    GOLDMAN, ME
    [J]. JOURNAL OF VIROLOGY, 1991, 65 (09) : 4887 - 4892
  • [35] POTENT AND SELECTIVE-INHIBITION OF HIV-1 REPLICATION INVITRO BY A NOVEL SERIES OF TIBO DERIVATIVES
    PAUWELS, R
    ANDRIES, K
    DESMYTER, J
    SCHOLS, D
    KUKLA, MJ
    BRESLIN, HJ
    RAEYMAECKERS, A
    VANGELDER, J
    WOESTENBORGHS, R
    HEYKANTS, J
    SCHELLEKENS, K
    JANSSEN, MAC
    DECLERCQ, E
    JANSSEN, PAJ
    [J]. NATURE, 1990, 343 (6257) : 470 - 474
  • [36] PAUWELS R, 1992, UNPUB ANTIMICROB AGE
  • [37] PAUWELS R, 1990, DESIGN ANTIAIDS DRUG, P103
  • [38] PAUWELS R, IN PRESS P NATL ACAD
  • [39] TSAO ANALOGS - STEREOSPECIFIC SYNTHESIS AND ANTI-HIV-1 ACTIVITY OF 1-[2',5'-BIS-0-(TERT-BUTYLDIMETHYLSILYL)-BETA-D-RIBOFURANOSYL]-3'-SPIRO-5''-(4''-AMINO-1'',2''-OXATHIOLE 2'',2''-DIOXIDE)PYRIMIDINE AND PYRIMIDINE-MODIFIED NUCLEOSIDES
    PEREZPEREZ, MJ
    SANFELIX, A
    BALZARINI, J
    DECLERCQ, E
    CAMARASA, MJ
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (16) : 2988 - 2995
  • [40] DIFFERENT PATTERN OF ACTIVITY OF INHIBITORS OF THE HUMAN-IMMUNODEFICIENCY-VIRUS IN LYMPHOCYTES AND MONOCYTE MACROPHAGES
    PERNO, CF
    YARCHOAN, R
    BALZARINI, J
    BERGAMINI, A
    MILANESE, G
    PAUWELS, R
    DECLERCQ, E
    ROCCHI, G
    CALIO, R
    [J]. ANTIVIRAL RESEARCH, 1992, 17 (04) : 289 - 304