STEREOSELECTIVE DELIVERY AND ACTIONS OF BETA-RECEPTOR-ANTAGONISTS

被引:137
作者
WALLE, T
WEBB, JG
BAGWELL, EE
WALLE, UK
DANIELL, HB
GAFFNEY, TE
机构
关键词
D O I
10.1016/0006-2952(88)90763-0
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:115 / 124
页数:10
相关论文
共 47 条
[1]   EFFECTS OF CANCER AND ITS TREATMENTS ON PLASMA-CONCENTRATION OF ALPHA-1-ACID GLYCOPROTEIN AND PROPRANOLOL BINDING [J].
ABRAMSON, FP ;
JENKINS, J ;
OSTCHEGA, Y .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1982, 32 (05) :659-663
[2]  
BAGWELL EE, 1986, 16TH SOC NEUR ANN M
[3]  
BAI SA, 1983, DRUG METAB DISPOS, V11, P394
[4]   GENETIC-POLYMORPHISM IN DRUG OXIDATION - INVITRO STUDIES OF HUMAN DEBRISOQUINE 4-HYDROXYLASE AND BUFURALOL 1'-HYDROXYLASE ACTIVITIES [J].
BOOBIS, AR ;
MURRAY, S ;
HAMPDEN, CE ;
DAVIES, DS .
BIOCHEMICAL PHARMACOLOGY, 1985, 34 (01) :65-71
[5]  
BORG KO, 1975, ACTA PHARMACOL TOX, V36, P125
[6]   DEPOLARIZATION-INDUCED RELEASE OF PROPRANOLOL AND ATENOLOL FROM RAT CORTICAL SYNAPTOSOMES [J].
BRIGHT, PS ;
GAFFNEY, TE ;
STREET, JA ;
WEBB, JG .
BRITISH JOURNAL OF PHARMACOLOGY, 1985, 84 (02) :499-510
[7]  
CHRIST DD, 1985, DRUG METAB DISPOS, V13, P380
[8]   PLASMA PROPRANOLOL LEVELS IN QUANTITATIVE ASSESSMENT OF BETA-ADRENERGIC BLOCKADE IN MAN [J].
COLTART, DJ ;
SHAND, DG .
BRITISH MEDICAL JOURNAL, 1970, 3 (5725) :731-&
[9]  
DANIELL HB, 1979, J PHARMACOL EXP THER, V208, P354
[10]   CHARACTERIZATION OF A COMMON GENETIC-DEFECT OF CYTOCHROME-P-450 FUNCTION (DEBRISOQUINE-SPARTEINE TYPE POLYMORPHISM) - INCREASED MICHAELIS CONSTANT (KM) AND LOSS OF STEREOSELECTIVITY OF BUFURALOL 1'-HYDROXYLATION IN POOR METABOLIZERS [J].
DAYER, P ;
GASSER, R ;
GUT, J ;
KRONBACH, T ;
ROBERTZ, GM ;
EICHELBAUM, M ;
MEYER, UA .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1984, 125 (01) :374-380