NEW PROGLUMIDE-ANALOG CCK RECEPTOR ANTAGONISTS - VERY POTENT AND SELECTIVE FOR PERIPHERAL-TISSUES

被引:17
作者
NIEDERAU, C
NIEDERAU, M
WILLIAMS, JA
GRENDELL, JH
机构
[1] UNIV CALIF SAN FRANCISCO,DEPT MED,SAN FRANCISCO,CA 94143
[2] UNIV CALIF SAN FRANCISCO,DEPT PHYSIOL,SAN FRANCISCO,CA 94143
[3] MT ZION HOSP & MED CTR,HAROLD BRUNN INST,CELL BIOL LAB,SAN FRANCISCO,CA 94120
来源
AMERICAN JOURNAL OF PHYSIOLOGY | 1986年 / 250卷 / 06期
关键词
D O I
10.1152/ajpgi.1986.250.6.G856
中图分类号
Q4 [生理学];
学科分类号
071003 ;
摘要
引用
收藏
页码:G856 / G860
页数:5
相关论文
共 26 条
[1]   CYCLIC-NUCLEOTIDE ANTAGONISTS OF CHOLECYSTOKININ - STRUCTURAL REQUIREMENTS FOR INTERACTION WITH THE CHOLECYSTOKININ RECEPTOR [J].
BARLAS, N ;
JENSEN, RT ;
BEINFELD, MC ;
GARDNER, JD .
AMERICAN JOURNAL OF PHYSIOLOGY, 1982, 242 (02) :G161-G167
[2]   LABELING OF PROTEINS TO HIGH SPECIFIC RADIOACTIVITIES BY CONJUGATION TO A I-125-CONTAINING ACYLATING AGENT - APPLICATION TO RADIOIMMUNOASSAY [J].
BOLTON, AE ;
HUNTER, WM .
BIOCHEMICAL JOURNAL, 1973, 133 (03) :529-538
[3]   A POTENT NONPEPTIDE CHOLECYSTOKININ ANTAGONIST SELECTIVE FOR PERIPHERAL-TISSUES ISOLATED FROM ASPERGILLUS-ALLIACEUS [J].
CHANG, RSL ;
LOTTI, VJ ;
MONAGHAN, RL ;
BIRNBAUM, J ;
STAPLEY, EO ;
GOETZ, MA ;
ALBERSSCHONBERG, G ;
PATCHETT, AA ;
LIESCH, JM ;
HENSENS, OD ;
SPRINGER, JP .
SCIENCE, 1985, 230 (4722) :177-179
[4]   PROGLUMIDE - SELECTIVE ANTAGONISM OF EXCITATORY EFFECTS OF CHOLECYSTOKININ IN CENTRAL NERVOUS-SYSTEM [J].
CHIODO, LA ;
BUNNEY, BS .
SCIENCE, 1983, 219 (4591) :1449-1450
[5]   DERIVATIVES OF CCK-(26-32) AS CHOLECYSTOKININ RECEPTOR ANTAGONISTS IN GUINEA-PIG PANCREATIC ACINI [J].
GARDNER, JD ;
KNIGHT, M ;
SUTLIFF, VE ;
TAMMINGA, CA ;
JENSEN, RT .
AMERICAN JOURNAL OF PHYSIOLOGY, 1984, 246 (03) :G292-G295
[6]   CHOLECYSTOKININ RECEPTOR ANTAGONISTS [J].
GARDNER, JD ;
JENSEN, RT .
AMERICAN JOURNAL OF PHYSIOLOGY, 1984, 246 (05) :G471-G476
[7]  
GRENDELL JH, 1985, GASTROENTEROLOGY, V88, P1405
[8]   PROGLUMIDE AND BENZOTRIPT - MEMBERS OF A DIFFERENT CLASS OF CHOLECYSTOKININ RECEPTOR ANTAGONISTS [J].
HAHNE, WF ;
JENSEN, RT ;
LEMP, GF ;
GARDNER, JD .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (10) :6304-6308
[9]   DISTINCT CHOLECYSTOKININ RECEPTORS IN BRAIN AND PANCREAS [J].
INNIS, RB ;
SNYDER, SH .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1980, 77 (11) :6917-6921
[10]   PROGLUMIDE ANALOGS - POTENT CHOLECYSTOKININ RECEPTOR ANTAGONISTS [J].
JENSEN, RT ;
MURPHY, RB ;
TRAMPOTA, M ;
SCHNEIDER, LH ;
JONES, SW ;
HOWARD, JM ;
GARDNER, JD .
AMERICAN JOURNAL OF PHYSIOLOGY, 1985, 249 (02) :G214-G220