CHRONIC BETA-ADRENOCEPTOR ANTAGONIST TREATMENT MODULATES HUMAN CARDIAC AND VASCULAR BETA-ADRENOCEPTOR DENSITY IN A SUBTYPE-SELECTIVE FASHION

被引:8
作者
BRODDE, OE [1 ]
MICHEL, MC [1 ]
WANG, XL [1 ]
ZERKOWSKI, HR [1 ]
机构
[1] UNIV ESSEN GESAMTHSCH,THORAX & KARDIOVASK CHIRURG ABT,D-4300 ESSEN 1,FED REP GER
关键词
D O I
10.1097/00004872-198812040-00157
中图分类号
R6 [外科学];
学科分类号
1002 ; 100210 ;
摘要
引用
收藏
页码:S497 / S500
页数:4
相关论文
共 19 条
[1]  
BOYUM A, 1968, SCAND J CLIN LAB INV, VS 21, P77
[2]   BETA-1-ADRENERGIC-RECEPTOR AND BETA-2-ADRENERGIC-RECEPTOR SUBPOPULATIONS IN NONFAILING AND FAILING HUMAN VENTRICULAR MYOCARDIUM - COUPLING OF BOTH RECEPTOR SUBTYPES TO MUSCLE-CONTRACTION AND SELECTIVE BETA-1-RECEPTOR DOWN-REGULATION IN HEART-FAILURE- [J].
BRISTOW, MR ;
GINSBURG, R ;
UMANS, V ;
FOWLER, M ;
MINOBE, W ;
RASMUSSEN, R ;
ZERA, P ;
MENLOVE, R ;
SHAH, P ;
JAMIESON, S ;
STINSON, EB .
CIRCULATION RESEARCH, 1986, 59 (03) :297-309
[3]   REGIONAL DISTRIBUTION OF BETA-ADRENOCEPTORS IN THE HUMAN-HEART - COEXISTENCE OF FUNCTIONAL BETA-1-ADRENOCEPTOR AND BETA-2-ADRENOCEPTOR IN BOTH ATRIA AND VENTRICLES IN SEVERE CONGESTIVE CARDIOMYOPATHY [J].
BRODDE, OE ;
SCHULER, S ;
KRETSCH, R ;
BRINKMANN, M ;
BORST, HG ;
HETZER, R ;
REIDEMEISTER, JC ;
WARNECKE, H ;
ZERKOWSKI, HR .
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY, 1986, 8 (06) :1235-1242
[4]   HUMAN-HEART BETA-ADRENOCEPTORS - A FAIR COMPARISON WITH LYMPHOCYTE BETA-ADRENOCEPTORS [J].
BRODDE, OE ;
BECKERINGH, JJ ;
MICHEL, MC .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1987, 8 (10) :403-407
[5]   BETA-ADRENOCEPTOR ANTAGONISTS (NONSELECTIVE AS WELL AS BETA-1-SELECTIVE) WITH PARTIAL AGONISTIC ACTIVITY DECREASE BETA-2-ADRENOCEPTOR DENSITY IN HUMAN-LYMPHOCYTES - EVIDENCE FOR A BETA-2-AGONISTIC COMPONENT OF THE PARTIAL AGONISTIC ACTIVIT [J].
BRODDE, OE ;
SCHEMUTH, R ;
BRINKMANN, M ;
WANG, XL ;
DAUL, A ;
BORCHARD, U .
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1986, 333 (02) :130-138
[6]   DIFFERENTIATION OF BETA-1-ADRENOCEPTOR AND BETA-2-ADRENOCEPTOR-MEDIATED EFFECTS IN HUMANS [J].
BRODDE, OE ;
DAUL, A ;
WELLSTEIN, A ;
PALM, D ;
MICHEL, MC ;
BECKERINGH, JJ .
AMERICAN JOURNAL OF PHYSIOLOGY, 1988, 254 (02) :H199-H206
[7]   TERBUTALINE-INDUCED DESENSITIZATION OF HUMAN-LYMPHOCYTE BETA-2-ADRENOCEPTORS - ACCELERATED RESTORATION OF BETA-ADRENOCEPTOR RESPONSIVENESS BY PREDNISONE AND KETOTIFEN [J].
BRODDE, OE ;
BRINKMANN, M ;
SCHEMUTH, R ;
OHARA, N ;
DAUL, A .
JOURNAL OF CLINICAL INVESTIGATION, 1985, 76 (03) :1096-1101
[8]  
BRODDE OE, 1988, IN PRESS ANN CLIN RE
[9]   ELEVATED BETA-ADRENERGIC-RECEPTOR NUMBER AFTER CHRONIC PROPRANOLOL TREATMENT [J].
GLAUBIGER, G ;
LEFKOWITZ, RJ .
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 1977, 78 (02) :720-725
[10]  
HEDBERG A, 1986, J PHARMACOL EXP THER, V239, P117