BETA-ADRENOCEPTOR ANTAGONISTS (NONSELECTIVE AS WELL AS BETA-1-SELECTIVE) WITH PARTIAL AGONISTIC ACTIVITY DECREASE BETA-2-ADRENOCEPTOR DENSITY IN HUMAN-LYMPHOCYTES - EVIDENCE FOR A BETA-2-AGONISTIC COMPONENT OF THE PARTIAL AGONISTIC ACTIVIT

被引:43
作者
BRODDE, OE [1 ]
SCHEMUTH, R [1 ]
BRINKMANN, M [1 ]
WANG, XL [1 ]
DAUL, A [1 ]
BORCHARD, U [1 ]
机构
[1] UNIV DUSSELDORF,INST PHARMACOL,D-4000 DUSSELDORF 1,FED REP GER
关键词
D O I
10.1007/BF00506515
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:130 / 138
页数:9
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共 40 条
  • [1] ELEVATION OF BETA-ADRENERGIC-RECEPTOR DENSITY IN HUMAN-LYMPHOCYTES AFTER PROPRANOLOL ADMINISTRATION
    AARONS, RD
    NIES, AS
    GAL, J
    HEGSTRAND, LR
    MOLINOFF, PB
    [J]. JOURNAL OF CLINICAL INVESTIGATION, 1980, 65 (05) : 949 - 957
  • [2] BORCHARD U, 1985, ARCH INT PHARMACOD T, V273, P4
  • [3] BOYUM A, 1968, SCAND J CLIN LAB INV, VS 21, P77
  • [4] EFFECTS OF BETA-ADRENOCEPTOR ANTAGONIST ADMINISTRATION ON BETA-2-ADRENOCEPTOR DENSITY IN HUMAN-LYMPHOCYTES - THE ROLE OF THE INTRINSIC SYMPATHOMIMETIC ACTIVITY
    BRODDE, OE
    DAUL, A
    STUKA, N
    OHARA, N
    BORCHARD, U
    [J]. NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY, 1985, 328 (04) : 417 - 422
  • [5] THE BETA-ADRENERGIC-RECEPTOR IN HUMAN-LYMPHOCYTES - SUBCLASSIFICATION BY THE USE OF A NEW RADIO-LIGAND, (+/-)-IODOCYANOPINDOLOL-125
    BRODDE, OE
    ENGEL, G
    HOYER, D
    BOCK, KD
    WEBER, F
    [J]. LIFE SCIENCES, 1981, 29 (21) : 2189 - 2198
  • [6] BRODDE OE, 1985, NAUNYNSCHMIEDE SR322, V329
  • [7] BRYAN LJ, 1981, J PHARMACOL EXP THER, V216, P395
  • [8] COMPARISON OF THE BETA-1-SELECTIVE AFFINITY OF PRENALTEROL AND CORWIN DEMONSTRATED BY RADIOLIGAND BINDING
    COOK, N
    RICHARDSON, A
    BARNETT, DB
    [J]. EUROPEAN JOURNAL OF PHARMACOLOGY, 1984, 98 (3-4) : 407 - 412
  • [9] COMPARISON OF THE CHRONOTROPIC EFFECT AND THE CYCLIC-AMP ACCUMULATION INDUCED BY BETA-2-AGONISTS IN RAT-HEART CELL-CULTURE
    FREYSSBEGUIN, M
    GRIFFATON, G
    LECHAT, P
    PICKEN, D
    QUENNEDEY, MC
    ROUOT, B
    SCHWARTZ, J
    [J]. BRITISH JOURNAL OF PHARMACOLOGY, 1983, 78 (04) : 717 - 723
  • [10] CONSTANT KINETICS AND CONSTANT CONCENTRATION-EFFECT RELATIONSHIP DURING LONG-TERM BETA-BLOCKADE WITH PINDOLOL
    GALEAZZI, RL
    PIROVINO, M
    WEIDMANN, P
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 1983, 33 (06) : 733 - 740