DEVELOPMENT OF A NEW PHYSICOCHEMICAL MODEL FOR BRAIN PENETRATION AND ITS APPLICATION TO THE DESIGN OF CENTRALLY ACTING H-2-RECEPTOR HISTAMINE-ANTAGONISTS

被引:477
作者
YOUNG, RC
MITCHELL, RC
BROWN, TH
GANELLIN, CR
GRIFFITHS, R
JONES, M
RANA, KK
SAUNDERS, D
SMITH, IR
SORE, NE
WILKS, TJ
机构
关键词
D O I
10.1021/jm00398a028
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
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页码:656 / 671
页数:16
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