TELENZEPINE IS AT LEAST 25 TIMES MORE POTENT THAN PIRENZEPINE - A DOSE-RESPONSE AND COMPARATIVE SECRETORY STUDY IN MAN

被引:33
作者
LONDONG, W [1 ]
LONDONG, V [1 ]
MEIERL, A [1 ]
VODERHOLZER, U [1 ]
机构
[1] UNIV MUNICH, MED KLIN, D-8000 MUNICH 2, GERMANY
关键词
D O I
10.1136/gut.28.7.888
中图分类号
R57 [消化系及腹部疾病];
学科分类号
摘要
引用
收藏
页码:888 / 895
页数:8
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共 30 条
[11]   CARDIOSELECTIVE PROFILE OF AF-DX-116, A MUSCARINE M2 RECEPTOR ANTAGONIST [J].
GIACHETTI, A ;
MICHELETTI, R ;
MONTAGNA, E .
LIFE SCIENCES, 1986, 38 (18) :1663-1672
[12]  
GILLARD BK, 1977, CLIN CHEM, V23, P2279
[13]  
HACKI WH, 1985, SCHWEIZ MED WSCHR, V115, P1033
[14]   BINDING PROFILE OF A NOVEL CARDIOSELECTIVE MUSCARINE RECEPTOR ANTAGONIST, AF-DX 116, TO MEMBRANES OF PERIPHERAL-TISSUES AND BRAIN IN THE RAT [J].
HAMMER, R ;
GIRALDO, E ;
SCHIAVI, GB ;
MONFERINI, E ;
LADINSKY, H .
LIFE SCIENCES, 1986, 38 (18) :1653-1662
[15]  
HAMMER R, 1977, THERAPIEWOCHE, V27, P1575
[16]  
JAUP BH, 1980, SCAND J GASTROENTERO, V15, P35
[17]  
KONTUREK SJ, 1980, SCAND J GASTROENTERO, V15, P63
[18]   SERUM GASTRIN AND GASTRIC-ACID RESPONSES TO MEALS AT VARIOUS PH LEVELS IN MAN [J].
KONTUREK, SJ ;
BIERNAT, J ;
OLEKSY, J .
GUT, 1974, 15 (07) :526-530
[19]  
LONDONG W, 1980, SCAND J GASTROENTERO, V15, P103
[20]   COMPLETE INHIBITION OF FOOD-STIMULATED GASTRIC-ACID SECRETION BY COMBINED APPLICATION OF PIRENZEPINE AND RANITIDINE [J].
LONDONG, W ;
LONDONG, V ;
RUTHE, C ;
WEIZERT, P .
GUT, 1981, 22 (07) :542-548