INHIBITION OF AROMATASE-ACTIVITY IN THE RAT BY AMINOGLUTETHIMIDE AND RELATED-COMPOUNDS

被引:7
作者
POURGHOLAMI, MH
NICHOLLS, PJ
SMITH, HJ
DALY, MJ
DYAS, J
机构
[1] UWIST,WELSH SCH PHARM,POB 13,CARDIFF CF1 3XF,WALES
[2] UNIV WALES COLL MED,TENOVUS INST CANC RES,CARDIFF CF4 4XX,S GLAM,WALES
关键词
D O I
10.1016/0022-4731(87)90094-X
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:309 / 312
页数:4
相关论文
共 28 条
[21]   ADRENAL SUPPRESSION WITH AMINOGLUTETHIMIDE .1. DIFFERENTIAL EFFECTS OF AMINOGLUTETHIMIDE ON GLUCOCORTICOID METABOLISM AS A RATIONALE FOR USE OF HYDROCORTISONE [J].
SANTEN, RJ ;
WELLS, SA ;
RUNIC, S ;
GUPTA, C ;
KENDALL, J ;
RUDY, EB ;
SAMOJLIK, E .
JOURNAL OF CLINICAL ENDOCRINOLOGY & METABOLISM, 1977, 45 (03) :469-479
[22]  
SANTEN RJ, 1982, CLIN ONCOLOGY, V1, P77
[23]   ESTROGEN FORMATION IN STROMAL CELLS OF ADIPOSE-TISSUE OF WOMEN - INDUCTION BY GLUCOCORTICOSTEROIDS [J].
SIMPSON, ER ;
ACKERMAN, GE ;
SMITH, ME ;
MENDELSON, CR .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA-BIOLOGICAL SCIENCES, 1981, 78 (09) :5690-5694
[24]   ENDOCRINE EFFECTS OF LOW-DOSE AMINOGLUTETHIMIDE AS AN AROMATASE INHIBITOR IN THE TREATMENT OF BREAST-CANCER [J].
STUARTHARRIS, R ;
DOWSETT, M ;
DSOUZA, A ;
DONALDSON, A ;
HARRIS, AL ;
JEFFCOATE, SL ;
SMITH, IE .
CLINICAL ENDOCRINOLOGY, 1985, 22 (02) :219-226
[25]  
THOMPSON EA, 1974, J BIOL CHEM, V249, P5373
[26]   AMINOGLUTETHIMIDE (WITH HYDROCORTISONE) INDUCED AGRANULOCYTOSIS IN PRIMARY BREAST-CANCER [J].
VINCENT, MD ;
CLINK, HM ;
COOMBES, RC ;
SMITH, IE ;
KANDLER, R ;
POWLES, TJ .
BRITISH MEDICAL JOURNAL, 1985, 291 (6488) :105-106
[27]  
WING LY, 1985, CANCER RES, V45, P2425
[28]  
ZIMNISKI SJ, 1985, CANCER RES, V45, P4883