BIOAVAILABILITY OF ORAL TRIMETREXATE IN PATIENTS WITH ACQUIRED IMMUNODEFICIENCY SYNDROME

被引:11
作者
ROGERS, P
ALLEGRA, CJ
MURPHY, RF
DRAKE, JC
MASUR, H
POPLACK, DG
CHABNER, BA
PARRILLO, JE
LANE, HC
BALIS, FM
机构
[1] NCI,PEDIAT BRANCH,BETHESDA,MD 20892
[2] NCI,CLIN PHARMACOL BRANCH,BETHESDA,MD 20892
[3] NCI,CTR CLIN,DEPT CRIT CARE MED,BETHESDA,MD 20892
关键词
D O I
10.1128/AAC.32.3.324
中图分类号
Q93 [微生物学];
学科分类号
071005 ; 100705 ;
摘要
引用
收藏
页码:324 / 326
页数:3
相关论文
共 16 条
  • [1] TRIMETREXATE FOR THE TREATMENT OF PNEUMOCYSTIS-CARINII PNEUMONIA IN PATIENTS WITH ACQUIRED-IMMUNODEFICIENCY-SYNDROME
    ALLEGRA, CJ
    CHABNER, BA
    TUAZON, CU
    OGATAARAKAKI, D
    BAIRD, B
    DRAKE, JC
    SIMMONS, JT
    LACK, EE
    SHELHAMER, JH
    BALIS, F
    WALKER, R
    KOVACS, JA
    LANE, HC
    MASUR, H
    [J]. NEW ENGLAND JOURNAL OF MEDICINE, 1987, 317 (16) : 978 - 985
  • [2] BALIS FM, 1987, CANCER RES, V47, P4973
  • [3] BALIS FM, 1983, CANCER RES, V43, P2342
  • [4] BALIS FM, 1986, CANCER RES, V46, P169
  • [5] 2,4-DIAMINO-5-METHYL-6-[(3,4,5-TRIMETHOXYANILINO)METHYL]QUINAZOLINE (TMQ), A POTENT NON-CLASSICAL FOLATE ANTAGONIST INHIBITOR .1. EFFECT ON DIHYDROFOLATE-REDUCTASE AND GROWTH OF RODENT TUMORS INVITRO AND INVIVO
    BERTINO, JR
    SAWICKI, WL
    MOROSON, BA
    CASHMORE, AR
    ELSLAGER, EF
    [J]. BIOCHEMICAL PHARMACOLOGY, 1979, 28 (12) : 1983 - 1987
  • [6] DIDDENS H, 1983, CANCER RES, V43, P5286
  • [7] Gibaldi M., 1982, PHARMACOKINETICS, P445
  • [8] HENDERSON ES, 1965, CANCER RES, V25, P1018
  • [9] CLINICAL-PHARMACOLOGY OF TRIMETREXATE
    HO, DHW
    COVINGTON, WP
    LEGHA, SS
    NEWMAN, RA
    KRAKOFF, IH
    [J]. CLINICAL PHARMACOLOGY & THERAPEUTICS, 1987, 42 (03) : 351 - 356
  • [10] UPTAKE AND EFFICACY OF TRIMETREXATE (TMQ, 2,4-DIAMINO-5-METHYL-6-[(3,4,5-TRIMETHOXYANILINO)METHYL] QUINAZOLINE), A NON-CLASSICAL ANTIFOLATE IN METHOTREXATE-RESISTANT LEUKEMIA-CELLS INVITRO
    KAMEN, BA
    EIBL, B
    CASHMORE, A
    BERTINO, J
    [J]. BIOCHEMICAL PHARMACOLOGY, 1984, 33 (10) : 1697 - 1699