Antivirals Targeting Influenza A Virus

被引:89
作者
Das, Kalyan [1 ]
机构
[1] Rutgers State Univ, Ctr Adv Biotechnol & Med, Dept Chem & Chem Biol, Piscataway, NJ 08854 USA
关键词
M2 PROTON CHANNELS; STRUCTURAL BASIS; RNA-POLYMERASE; ACTIVE-SITE; IN-VITRO; NEURAMINIDASE INHIBITORS; CRYSTAL-STRUCTURE; CAP-BINDING; ION-CHANNEL; AMINO-ACID;
D O I
10.1021/jm300455c
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:6263 / 6277
页数:15
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共 152 条
[1]   Structure and mechanism of proton transport through the transmembrane tetrameric M2 protein bundle of the influenza A virus [J].
Acharya, Rudresh ;
Carnevale, Vincenzo ;
Fiorin, Giacomo ;
Levine, Benjamin G. ;
Polishchuk, Alexei L. ;
Balannik, Victoria ;
Samish, Ilan ;
Lamb, Robert A. ;
Pinto, Lawrence H. ;
DeGrado, William F. ;
Klein, Michael L. .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2010, 107 (34) :15075-15080
[2]   Remarkable loop flexibility in avian influenza N1 and its implications for antiviral drug design [J].
Amaro, Rommie E. ;
Minh, David D. L. ;
Cheng, Lily S. ;
Lindstrom, William M., Jr. ;
Olson, Arthur J. ;
Lin, Jung-Hsin ;
Li, Wilfred W. ;
McCammon, J. Andrew .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2007, 129 (25) :7764-+
[3]   Mechanism of 150-cavity formation in influenza neuraminidase [J].
Amaro, Rommie E. ;
Swift, Robert V. ;
Votapka, Lane ;
Li, Wilfred W. ;
Walker, Ross C. ;
Bush, Robin M. .
NATURE COMMUNICATIONS, 2011, 2
[4]   3D structure of the influenza virus polymerase complex:: Localization of subunit domains [J].
Area, E ;
Martín-Benito, J ;
Gastaminza, P ;
Torreira, E ;
Valpuesta, JM ;
Carrascosa, JL ;
Ortín, J .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2004, 101 (01) :308-313
[5]   Functional Studies and Modeling of Pore-Lining Residue Mutants of the Influenza A Virus M2 Ion Channel [J].
Balannik, Victoria ;
Carnevale, Vincenzo ;
Fiorin, Giacomo ;
Levine, Benjamin G. ;
Lamb, Robert A. ;
Klein, Michael L. ;
DeGrado, William F. ;
Pinto, Lawrence H. .
BIOCHEMISTRY, 2010, 49 (04) :696-708
[6]   Anti-influenza virus activity of peramivir in mice with single intramuscular injection [J].
Bantia, S ;
Arnold, CS ;
Parker, CD ;
Upshaw, R ;
Chand, P .
ANTIVIRAL RESEARCH, 2006, 69 (01) :39-45
[7]   Epidemiological, antigenic and genetic characteristics of seasonal influenza A(H1N1), A(H3N2) and B influenza viruses: Basis for the WHO recommendation on the composition of influenza vaccines for use in the 2009-2010 Northern Hemisphere season [J].
Barr, Ian G. ;
McCauley, John ;
Cox, Nancy ;
Daniels, Rod ;
Engelhardt, Othmar G. ;
Fukuda, Keiji ;
Grohmann, Gary ;
Hay, Alan ;
Kelso, Anne ;
Klimov, Alexander ;
Odagiri, Takato ;
Smith, Derek ;
Russell, Colin ;
Tashiro, Masato ;
Webby, Richard ;
Wood, John ;
Ye, Zhiping ;
Zhang, Wenqing .
VACCINE, 2010, 28 (05) :1156-1167
[8]   Identification of Influenza Endonuclease Inhibitors Using a Novel Fluorescence Polarization Assay [J].
Baughman, Brandi M. ;
Slavish, P. Jake ;
DuBois, Rebecca M. ;
Boyd, Vincent A. ;
White, Stephen W. ;
Webb, Thomas R. .
ACS CHEMICAL BIOLOGY, 2012, 7 (03) :526-534
[9]   STRUCTURAL BASIS FOR THE 3'-5' EXONUCLEASE ACTIVITY OF ESCHERICHIA-COLI DNA-POLYMERASE-I - A 2 METAL-ION MECHANISM [J].
BEESE, LS ;
STEITZ, TA .
EMBO JOURNAL, 1991, 10 (01) :25-33
[10]   The Emergency Use Authorization of Peramivir for Treatment of 2009 H1N1 Influenza [J].
Birnkrant, Debra ;
Cox, Edward .
NEW ENGLAND JOURNAL OF MEDICINE, 2009, 361 (23) :2204-2207