Lithium perchlorate assisted one-pot three-component aminoalkylation of electron-rich aromatic compounds

被引：71

作者：

Saidi, MR ^{[1
]}

Azizi, N ^{[1
]}

Naimi-Jamal, MR ^{[1
]}

机构：

[1] Sharif Univ Technol, Dept Chem, Tehran, Iran

来源：

TETRAHEDRON LETTERS | 2001年 / 42卷 / 45期

关键词：

aminoalkylation; Mannich reaction; lithium perchlorate; electron-rich aromatic compounds;

D O I：

10.1016/S0040-4039(01)01732-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A one-pot. three-component. Mannich reaction of electron-rich aromatic compounds with in situ prepared iminium salts in 5 M ethereal lithium perchlorate gives good yields of aminoalkylated products at room temperature. (C) 2001 Elsevier Science Ltd. All rights reserved.

引用

页码：8111 / 8113

页数：3

共 18 条

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