A very short, efficient and inexpensive synthesis of the prodrug form of SC-54701A - A platelet aggregation inhibitor

被引：22

作者：

Cossy, J ^{[1
]}

Schmitt, A ^{[1
]}

Cinquin, C ^{[1
]}

Buisson, D ^{[1
]}

Belotti, D ^{[1
]}

机构：

[1] UNIV PARIS 05,CHIM & BIOCHIM PHARMACOL & TOXICOL LAB,CNRS,F-75270 PARIS 06,FRANCE

来源：

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS | 1997年 / 7卷 / 13期

关键词：

D O I：

10.1016/S0960-894X(97)00293-X

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

A short and efficient synthesis of the prodrug form of SC-54701A has been achieved from (trimethylsilyl)acetylene in 6 steps with an overall yield of 19%. (C) 1997 Elsevier Science Ltd.

引用

收藏

页码：1699 / 1700

页数：2

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