A convenient synthesis of beta-acyl glucuronides

被引：39

作者：

Juteau, H

Gareau, Y

Labelle, M

机构：

[1] Merck Frosst Ctr. Therapeut. Res., Pointe-Claire-Dorval, Que. H9R 4P8

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 09期

关键词：

D O I：

10.1016/S0040-4039(97)00135-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

引用

页码：1481 / 1484

页数：4

共 19 条

[1]

[Anonymous], 1960, UNIVERSITAS, V4, P397

[2]

BEAUPERE D, 1994, TETRAHEDRON LETT, V35, P6279

[3] CHEMICAL SYNTHESIS OF I-O-INDOMETHACIN-BETA-D-GLUCOSYLURONIC ACID [J].

BUGIANESI, R ;

SHEN, TY .

CARBOHYDRATE RESEARCH, 1971, 19 (02) :179-+

[4] A NEW PROTECTED FORM OF GLUCURONIC-ACID FOR THE SYNTHESIS OF LABILE 1-O-ACYL-BETA-D-GLUCURONIDES [J].

DEMESMAEKER, A ;

HOFFMANN, P ;

ERNST, B .

TETRAHEDRON LETTERS, 1989, 30 (29) :3773-3776

[5]

Dutton GJ, 1980, GLUCURONIDATION DRUG

[6] SOLID-PHASE SYNTHESIS OF DRUG GLUCURONIDES BY IMMOBILIZED GLUCURONOSYLTRANSFERASE [J].

FENSELAU, C ;

PALLANTE, S ;

PARIKH, I .

JOURNAL OF MEDICINAL CHEMISTRY, 1976, 19 (05) :679-683

[7] ISOLATION AND IDENTIFICATION OF THE REARRANGEMENT PRODUCTS OF DIFLUNISAL 1-O-ACYL GLUCURONIDE [J].

HANSENMOLLER, J ;

CORNETT, C ;

DALGAARD, L ;

HANSEN, SH .

JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 1988, 6 (03) :229-240

[8]

Hughes D.L., 1992, ORG REACT, V42, P335, DOI [10.1002/0471264180.OR042.02, DOI 10.1002/0471264180.OR042.02]

[9] The effect of acid strength on the Mitsunobu esterification reaction: Carboxyl vs hydroxyl reactivity [J].

Hughes, DL ;

Reamer, RA .

JOURNAL OF ORGANIC CHEMISTRY, 1996, 61 (09) :2967-2971

[10] DISCOVERY OF MK-0476, A POTENT AND ORALLY-ACTIVE LEUKOTRIENE D-4 RECEPTOR ANTAGONIST DEVOID OF PEROXISOMAL ENZYME-INDUCTION [J].

LABELLE, M ;

BELLEY, M ;

GAREAU, Y ;

GAUTHIER, JY ;

GUAY, D ;

GORDON, R ;

GROSSMAN, SG ;

JONES, TR ;

LEBLANC, Y ;

MCAULIFFE, M ;

MCFARLANE, C ;

MASSON, P ;

METTERS, KM ;

OUIMET, N ;

PATRICK, DH ;

PIECHUTA, H ;

ROCHETTE, C ;

SAWYER, N ;

XIANG, YB ;

PICKETT, CB ;

FORDHUTCHINSON, AW ;

ZAMBONI, RJ ;

YOUNG, RN .

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1995, 5 (03) :283-288

← 1 2 →