Synthesis of 1,2,3-Trisubstituted pyrrolo[3,2-c]quinolines via palladium-catalyzed heteroannulation with internal alkynes

被引：52

作者：

Kang, SK ^{[1
]}

Park, SS ^{[1
]}

Kim, SS ^{[1
]}

Choi, JK ^{[1
]}

Yum, EK ^{[1
]}

机构：

[1] Korea Res Inst Chem Technol, Bioorgan Sci Div, Taejon 305600, South Korea

来源：

TETRAHEDRON LETTERS | 1999年 / 40卷 / 23期

关键词：

D O I：

10.1016/S0040-4039(99)00753-4

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Various 1,2,3-trisubstituted pyrrolo[3,2-c]quinolines were synthesized by palladium-catalyzed heteroannulation of 4-amino-3-iodoquinoline derivatives and internal alkynes. The 1,2,3-trisubstituted pyrrolo[3,2-c]quinolines could be further transformed by desilylation, debenzylation, or substitution. (C) 1999 Elsevier Science Ltd. All rights reserved.

引用

页码：4379 / 4382

页数：4

共 24 条

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