Novel A,B,E-ring-modified camptothecins displaying high lipophilicity and markedly improved human blood stabilities

被引：68

作者：

Bom, D

Curran, DP

Chavan, AJ

Kruszewski, S

Zimmer, SG

Fraley, KA

Burke, TG

机构：

[1] Univ Kentucky, Coll Pharm, Div Pharmaceut Sci, Lexington, KY 40506 USA

[2] Univ Pittsburgh, Dept Chem, Pittsburgh, PA 15260 USA

[3] Tigen Pharmaceut Inc, Lexington, KY 40506 USA

[4] Univ Kentucky, Coll Med, Dept Microbiol & Immunol, Lexington, KY 40506 USA

[5] Univ Kentucky, Lucille P Markey Canc Ctr, Lexington, KY 40506 USA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1999年 / 42卷 / 16期

关键词：

D O I：

10.1021/jm9902279

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

引用

页码：3018 / 3022

页数：5

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