Orally active squalene synthase inhibitors: Bis((acyloxy)alkyl) prodrugs of the alpha-phosphonosulfonic acid moiety

被引：52

作者：

Dickson, JK

Biller, SA

Magnin, DR

Petrillo, EW

Hillyer, JW

Hsieh, DC

Lan, SJ

Rinehart, JK

Gregg, RE

Harrity, TW

Jolibois, KG

Kalinowski, SS

Kunselman, LK

Mookhtiar, KA

Ciosek, CP

机构：

[1] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DIV DISCOVERY CHEM,PRINCETON,NJ 08543

[2] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT METAB & PHARMACOKINET,PRINCETON,NJ 08543

[3] BRISTOL MYERS SQUIBB PHARMACEUT RES INST,DEPT METAB DIS,PRINCETON,NJ 08543

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1996年 / 39卷 / 03期

关键词：

D O I：

10.1021/jm950735s

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：661 / 664

页数：4

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