Synthesis of 1′-β-D-glucopyranosyl-1,2,3-triazole-4,5-dimethanol-4,5-bis-(isopropylcarbamate) as potential antineoplastic agent

被引：69

作者：

Al-Masoudi, NA

Al-Soud, YA

机构：

[1] Univ Konstanz, Fak Chem, D-78457 Constance, Germany

[2] Univ Al Al Bayt, Coll Sci, Dept Chem, Al Mafraq, Jordan

来源：

TETRAHEDRON LETTERS | 2002年 / 43卷 / 22期

关键词：

D O I：

10.1016/S0040-4039(02)00733-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The title compound 5 was prepared from the I-P-D-azido-glucose I via four steps. Alternatively, 5 was synthesized from 1, via acetalation, cycloaddition with acetylene derivative, reduction, then carbamoylation followed by an acid hydrolysis. (C) 2002 Elsevier Science Ltd. All rights reserved.

引用

页码：4021 / 4022

页数：2

共 6 条

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