Reactivity as glycine templates of 1,2-dialkyl-2,4-dihydro-1H-pyrazino[2,1-b]quinazoline-3,6-diones

被引：13

作者：

Buenadicha, FL ^{[1
]}

Avendaño, C ^{[1
]}

Söllhuber, M ^{[1
]}

机构：

[1] Univ Complutense, Dept Quim Organ & Farmaceut, E-28040 Madrid, Spain

来源：

TETRAHEDRON-ASYMMETRY | 2001年 / 12卷 / 21期

关键词：

D O I：

10.1016/S0957-4166(01)00515-8

中图分类号：

O61 [无机化学];

学科分类号：

070301 ; 081704 ;

摘要：

The 1-methyl(iso-propyl)-2-benzyl-2,4-dihydro-1H-pyrazino[2,1-b]quinazoline-3,6-diones 8 and 9 could be regio- and diastereoselectively alkylated at C(4) with retention of configuration at both stereocentres. (C) 2002 Elsevier Science Ltd. All rights reserved.

引用

页码：3019 / 3028

页数：10

共 21 条

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