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Ras farnesyltransferase inhibitors
被引:22
作者
:
AyralKaloustian, S
论文数:
0
引用数:
0
h-index:
0
机构:
Wyeth-Ayerst Research, Pearl River
AyralKaloustian, S
Skotnicki, JS
论文数:
0
引用数:
0
h-index:
0
机构:
Wyeth-Ayerst Research, Pearl River
Skotnicki, JS
机构
:
[1]
Wyeth-Ayerst Research, Pearl River
来源
:
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 31
|
1996年
/ 31卷
关键词
:
D O I
:
10.1016/S0065-7743(08)60457-1
中图分类号
:
R9 [药学];
学科分类号
:
1007 ;
摘要
:
[No abstract available]
引用
收藏
页码:171 / 180
页数:10
相关论文
共 80 条
[1]
AOKI K, 1995, CANCER RES, V55, P3810
[2]
RATIONAL DESIGN OF POTENT CARBOXYLIC-ACID BASED BISUBSTRATE INHIBITORS OF RAS FARNESYL-PROTEIN TRANSFERASE
BHIDE, RS
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
BHIDE, RS
PATEL, DV
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
PATEL, DV
PATEL, MM
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
PATEL, MM
ROBINSON, SP
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
ROBINSON, SP
HUNIHAN, LW
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
HUNIHAN, LW
GORDON, EM
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
GORDON, EM
[J].
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1994,
4
(17)
: 2107
-
2112
[3]
Novel tricyclic inhibitors of farnesyl protein transferase - Biochemical characterization and inhibition of Ras modification in transfected Cos cells
Bishop, WR
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Bishop, WR
Bond, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Bond, R
Petrin, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Petrin, J
Wang, L
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Wang, L
Patton, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Patton, R
Doll, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Doll, R
Njoroge, G
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Njoroge, G
Catino, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Catino, J
Schwartz, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Schwartz, J
Windsor, W
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Windsor, W
Syto, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Syto, R
Schwartz, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Schwartz, J
Carr, D
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Carr, D
James, L
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
James, L
Kirschmeier, P
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Kirschmeier, P
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1995,
270
(51)
: 30611
-
30618
[4]
BOLTON GL, 1994, ANNU REP MED CHEM, V29, P165
[5]
BOS JL, 1989, CANCER RES, V49, P4682
[6]
BUSS BE, 1995, CHEM BIOL, V2, P787
[7]
LOCAL CONSTRAINED SHIFTY PSEUDOPEPTIDES INHIBITORS OF RAS-FARNESYL TRANSFERASE
BYK, G
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
BYK, G
DUCHESNE, M
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DUCHESNE, M
PARKER, F
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
PARKER, F
LELIEVRE, Y
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
LELIEVRE, Y
GUITTON, JD
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
GUITTON, JD
CLERC, FF
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
CLERC, FF
BECQUART, J
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
BECQUART, J
TOCQUE, B
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
TOCQUE, B
SCHERMAN, D
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
SCHERMAN, D
[J].
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1995,
5
(22)
: 2677
-
2682
[8]
CASEY PJ, 1996, IN PRESS J BIOL CHEM, V271
[9]
Phosphorylation of Bcl-2 protein and association with p21(Ras) in Ras-induced apoptosis
Chen, CY
论文数:
0
引用数:
0
h-index:
0
机构:
BOSTON UNIV,SCH MED,CTR CANC RES,BOSTON,MA 02118
Chen, CY
Faller, DV
论文数:
0
引用数:
0
h-index:
0
机构:
BOSTON UNIV,SCH MED,CTR CANC RES,BOSTON,MA 02118
Faller, DV
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1996,
271
(05)
: 2376
-
2379
[10]
CONSTRAINED ANALOGS OF KCVFM WITH IMPROVED INHIBITORY PROPERTIES AGAINST FARNESYL TRANSFERASE
CLERC, FF
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
CLERC, FF
GUITTON, JD
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
GUITTON, JD
FROMAGE, N
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
FROMAGE, N
LELIEVRE, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
LELIEVRE, Y
DUCHESNE, M
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
DUCHESNE, M
TOCQUE, B
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
TOCQUE, B
JAMESSURCOUF, E
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
JAMESSURCOUF, E
COMMERCON, A
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
COMMERCON, A
BECQUART, J
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
BECQUART, J
[J].
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1995,
5
(16)
: 1779
-
1784
←
1
2
3
4
5
6
7
8
→
共 80 条
[1]
AOKI K, 1995, CANCER RES, V55, P3810
[2]
RATIONAL DESIGN OF POTENT CARBOXYLIC-ACID BASED BISUBSTRATE INHIBITORS OF RAS FARNESYL-PROTEIN TRANSFERASE
BHIDE, RS
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
BHIDE, RS
PATEL, DV
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
PATEL, DV
PATEL, MM
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
PATEL, MM
ROBINSON, SP
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
ROBINSON, SP
HUNIHAN, LW
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
HUNIHAN, LW
GORDON, EM
论文数:
0
引用数:
0
h-index:
0
机构:
Bristol-Myers Squibb Pharmaceutical Research Institute, Princeton
GORDON, EM
[J].
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1994,
4
(17)
: 2107
-
2112
[3]
Novel tricyclic inhibitors of farnesyl protein transferase - Biochemical characterization and inhibition of Ras modification in transfected Cos cells
Bishop, WR
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Bishop, WR
Bond, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Bond, R
Petrin, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Petrin, J
Wang, L
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Wang, L
Patton, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Patton, R
Doll, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Doll, R
Njoroge, G
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Njoroge, G
Catino, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Catino, J
Schwartz, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Schwartz, J
Windsor, W
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Windsor, W
Syto, R
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Syto, R
Schwartz, J
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Schwartz, J
Carr, D
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Carr, D
James, L
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
James, L
Kirschmeier, P
论文数:
0
引用数:
0
h-index:
0
机构:
SCHERING PLOUGH CORP,RES INST,DEPT STRUCT CHEM,KENILWORTH,NJ 07033
Kirschmeier, P
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1995,
270
(51)
: 30611
-
30618
[4]
BOLTON GL, 1994, ANNU REP MED CHEM, V29, P165
[5]
BOS JL, 1989, CANCER RES, V49, P4682
[6]
BUSS BE, 1995, CHEM BIOL, V2, P787
[7]
LOCAL CONSTRAINED SHIFTY PSEUDOPEPTIDES INHIBITORS OF RAS-FARNESYL TRANSFERASE
BYK, G
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
BYK, G
DUCHESNE, M
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DUCHESNE, M
PARKER, F
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
PARKER, F
LELIEVRE, Y
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
LELIEVRE, Y
GUITTON, JD
论文数:
0
引用数:
0
h-index:
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机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
GUITTON, JD
CLERC, FF
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
CLERC, FF
BECQUART, J
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
BECQUART, J
TOCQUE, B
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
TOCQUE, B
SCHERMAN, D
论文数:
0
引用数:
0
h-index:
0
机构:
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
DEPT BIOTECHNOL, F-94403 VITRY, FRANCE
SCHERMAN, D
[J].
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1995,
5
(22)
: 2677
-
2682
[8]
CASEY PJ, 1996, IN PRESS J BIOL CHEM, V271
[9]
Phosphorylation of Bcl-2 protein and association with p21(Ras) in Ras-induced apoptosis
Chen, CY
论文数:
0
引用数:
0
h-index:
0
机构:
BOSTON UNIV,SCH MED,CTR CANC RES,BOSTON,MA 02118
Chen, CY
Faller, DV
论文数:
0
引用数:
0
h-index:
0
机构:
BOSTON UNIV,SCH MED,CTR CANC RES,BOSTON,MA 02118
Faller, DV
[J].
JOURNAL OF BIOLOGICAL CHEMISTRY,
1996,
271
(05)
: 2376
-
2379
[10]
CONSTRAINED ANALOGS OF KCVFM WITH IMPROVED INHIBITORY PROPERTIES AGAINST FARNESYL TRANSFERASE
CLERC, FF
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
CLERC, FF
GUITTON, JD
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
GUITTON, JD
FROMAGE, N
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
FROMAGE, N
LELIEVRE, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
LELIEVRE, Y
DUCHESNE, M
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
DUCHESNE, M
TOCQUE, B
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
TOCQUE, B
JAMESSURCOUF, E
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
JAMESSURCOUF, E
COMMERCON, A
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
COMMERCON, A
BECQUART, J
论文数:
0
引用数:
0
h-index:
0
机构:
Rhône-Poulenc Rorer S.A.- Centre de Recherches de Vitry-Alfortville 13, 94403 Vitry-sur-Seine
BECQUART, J
[J].
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
1995,
5
(16)
: 1779
-
1784
←
1
2
3
4
5
6
7
8
→