Ras farnesyltransferase inhibitors

被引:22
作者
AyralKaloustian, S
Skotnicki, JS
机构
[1] Wyeth-Ayerst Research, Pearl River
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 31 | 1996年 / 31卷
关键词
D O I
10.1016/S0065-7743(08)60457-1
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:171 / 180
页数:10
相关论文
共 80 条
  • [11] DALTON MB, 1995, CANCER RES, V55, P3295
  • [12] PSEUDODIPEPTIDE INHIBITORS OF PROTEIN FARNESYLTRANSFERASE
    DESOLMS, SJ
    DEANA, AA
    GIULIANI, EA
    GRAHAM, SL
    KOHL, NE
    MOSSER, SD
    OLIFF, AI
    POMPLIANO, DL
    RANDS, E
    SCHOLZ, TH
    WIGGINS, JM
    GIBBS, JB
    SMITH, RL
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 1995, 38 (20) : 3967 - 3971
  • [13] DESOLMS SJ, 1996, Patent No. 5491164
  • [14] DESOLMS SJ, 1995, Patent No. 5468733
  • [15] DESOLMS SJ, 1995, Patent No. 5439918
  • [16] Yeast protein farnesyltransferase: Steady-state kinetic studies of substrate binding
    Dolence, JM
    Cassidy, PB
    Mathis, JR
    Poulter, CD
    [J]. BIOCHEMISTRY, 1995, 34 (51) : 16687 - 16694
  • [17] PROTEIN FARNESYLTRANSFERASE - KINETICS OF FARNESYL PYROPHOSPHATE BINDING AND PRODUCT RELEASE
    FURFINE, ES
    LEBAN, JJ
    LANDAVAZO, A
    MOOMAW, JF
    CASEY, PJ
    [J]. BIOCHEMISTRY, 1995, 34 (20) : 6857 - 6862
  • [18] FARNESYLTRANSFERASE INHIBITORS - RAS RESEARCH YIELDS A POTENTIAL CANCER THERAPEUTIC
    GIBBS, JB
    OLIFF, A
    KOHL, NE
    [J]. CELL, 1994, 77 (02) : 175 - 178
  • [19] GIBBS JB, 1995, Patent No. 9520396
  • [20] GRAHAM SL, 1995, Patent No. 9500497