High-resolution X-ray crystallography reveals precise binding interactions between human nonpancreatic secreted phospholipase A(2) and a highly potent inhibitor (FPL67047XX)

被引：36

作者：

Cha, SS

Lee, D

Adams, J

Kurdyla, JT

Jones, CS

Marshall, LA

Bolognese, B

AbdelMeguid, SS

Oh, BH

机构：

[1] SMITHKLINE BEECHAM PHARMACEUT, DEPT MACROMOL SCI, KING OF PRUSSIA, PA 19406 USA

[2] SMITHKLINE BEECHAM PHARMACEUT, DEPT MED CHEM, KING OF PRUSSIA, PA 19406 USA

[3] SMITHKLINE BEECHAM PHARMACEUT, DEPT BIOCHEM, KING OF PRUSSIA, PA 19406 USA

[4] SMITHKLINE BEECHAM PHARMACEUT, DEPT INFLAMMAT & RESP PHARMACOL, KING OF PRUSSIA, PA 19406 USA

[5] POHANG UNIV SCI & TECHNOL, DEPT LIFE SCI, KYUNGBUK 790784, SOUTH KOREA

来源：

JOURNAL OF MEDICINAL CHEMISTRY | 1996年 / 39卷 / 20期

关键词：

D O I：

10.1021/jm960502g

中图分类号：

R914 [药物化学];

学科分类号：

100701 ;

摘要：

[No abstract available]

引用

页码：3878 / 3881

页数：4

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