Mechanism of action of p-glycoprotein in relation to passive membrane permeation

被引:65
作者
Eytan, GD [1 ]
Kuchel, PW
机构
[1] Technion Israel Inst Technol, Dept Biol, IL-32000 Haifa, Israel
[2] Univ Sydney, Dept Biochem, Sydney, NSW 2006, Australia
来源
INTERNATIONAL REVIEW OF CYTOLOGY - A SURVEY OF CELL BIOLOGY, VOL 190 | 1999年 / 190卷
关键词
p-glycoprotein; multidrug resistance; flip-flop; transmembrane movement; ABC transporter;
D O I
10.1016/S0074-7696(08)62148-8
中图分类号
Q2 [细胞生物学];
学科分类号
071009 ; 090102 ;
摘要
引用
收藏
页码:175 / 250
页数:76
相关论文
共 186 条
[11]   KINETIC-ANALYSIS OF CARRIER-MEDIATED ION-TRANSPORT BY CHARGE-PULSE TECHNIQUE [J].
BENZ, R ;
LAUGER, P .
JOURNAL OF MEMBRANE BIOLOGY, 1976, 27 (1-2) :171-191
[12]  
BERTHON HA, 1995, ADV MOL CELL BIOL, P147
[13]   RECONSTITUTION OF A BACTERIAL PERIPLASMIC PERMEASE IN PROTEOLIPOSOMES AND DEMONSTRATION OF ATP HYDROLYSIS CONCOMITANT WITH TRANSPORT [J].
BISHOP, L ;
AGBAYANI, R ;
AMBUDKAR, SV ;
MALONEY, PC ;
AMES, GFL .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1989, 86 (18) :6953-6957
[14]  
BOESCH D, 1991, CANCER RES, V51, P4226
[15]   Multidrug resistance in Lactococcus lactis: Evidence for ATP-dependent drug extrusion from the inner leaflet of the cytoplasmic membrane [J].
Bolhuis, H ;
vanVeen, HW ;
Molenaar, D ;
Poolman, B ;
Driessen, AJM ;
Konings, WN .
EMBO JOURNAL, 1996, 15 (16) :4239-4245
[16]   Competition of hydrophobic peptides, cytotoxic drugs, and chemosensitizers on a common P-glycoprotein pharmacophore as revealed by its ATPase activity [J].
Borgnia, MJ ;
Eytan, GD ;
Assaraf, YG .
JOURNAL OF BIOLOGICAL CHEMISTRY, 1996, 271 (06) :3163-3171
[17]   ANALYSIS OF DRUG TRANSPORT KINETICS IN MULTIDRUG-RESISTANT CELLS USING A NOVEL COUMARIN-VINBLASTINE COMPOUND [J].
BORNMANN, WG ;
ROEPE, PD .
BIOCHEMISTRY, 1994, 33 (42) :12665-12675
[18]   MOBILE IONOPHORES ARE A NOVEL CLASS OF P-GLYCOPROTEIN INHIBITORS - THE EFFECTS OF IONOPHORES ON 4'-O-TETRAHYDROPYRANYL-ADRIAMYCIN INCORPORATION IN K562 DRUG-RESISTANT CELLS [J].
BORREL, MN ;
PEREIRA, E ;
FIALLO, M ;
GARNIERSUILLEROT, A .
EUROPEAN JOURNAL OF BIOCHEMISTRY, 1994, 223 (01) :125-133
[19]   THE BLOOD-BRAIN-BARRIER - TRANSPORT ACROSS THE CEREBRAL ENDOTHELIUM [J].
BRADBURY, MWB .
CIRCULATION RESEARCH, 1985, 57 (02) :213-222
[20]   MECHANISM OF MULTIDRUG RESISTANCE [J].
BRADLEY, G ;
JURANKA, PF ;
LING, V .
BIOCHIMICA ET BIOPHYSICA ACTA, 1988, 948 (01) :87-128