Microwave-promoted transformations: Fast and chemoselective N-acylation of amino alcohols using catalytic amounts of dibutyltin oxide. Influence of the power output and the nature of the acylating agent on the selectivity

被引：52

作者：

Morcuende, A ^{[1
]}

Ors, M ^{[1
]}

Valverde, S ^{[1
]}

Herradon, B ^{[1
]}

机构：

[1] CSIC,INST QUIM ORGAN GEN,E-28006 MADRID,SPAIN

来源：

JOURNAL OF ORGANIC CHEMISTRY | 1996年 / 61卷 / 16期

关键词：

D O I：

10.1021/jo9605511

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The influence of the nature of the acylating agent and the power output on the chemoselectivity of the microwave-mediated acylation of 1,2- and 1,3-amino alcohols catalyzed by dibutyltin oxide has been studied. The method constitutes an efficient procedure for the selective N-acylation of amino alcohols.

引用

页码：5264 / 5270

页数：7

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