GABA(A) receptor pharmacology

被引:265
作者
Johnston, GAR
机构
关键词
GABA receptors; bicuculline; barbiturates; benzodiazepines; neuroactive steroids;
D O I
10.1016/0163-7258(95)02043-8
中图分类号
R9 [药学];
学科分类号
1007 [药学];
摘要
gamma-Aminobutyric acid (GABA)(A) receptors for the inhibitory neurotransmitter GABA are likely to be found on most, if not all, neurons in the brain and spinal cord, They appear to be the most complicated of the superfamily of ligand-gated ion channels in terms of the large number of receptor subtypes and also the variety of ligands that interact with specific sites on the receptors. There appear to be at least 11 distinct sites on GABA(A) receptors for these ligands.
引用
收藏
页码:173 / 198
页数:26
相关论文
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