Regiospecific and enantioselective synthesis of methylated metabolites of tea catechins

被引:47
作者
Wan, Sheng Biao
Dou, Q. Ping
Chan, Tak Hang [1 ]
机构
[1] Hong Kong Polytech Univ, Inst Mol Technol Drug Discovery & Synth, Dept Appl Biol, Kowloon, Hong Kong, Peoples R China
[2] Hong Kong Polytech Univ, Inst Mol Technol Drug Discovery & Synth, State Key Lab Chinese Med & Mol Pharmacol, Kowloon, Hong Kong, Peoples R China
[3] Wayne State Univ, Sch Med, Barbara Ann Karmanos Canc Inst, Prevent Program, Detroit, MI 48202 USA
[4] Wayne State Univ, Sch Med, Dept Pathol, Detroit, MI 48202 USA
关键词
D O I
10.1016/j.tet.2006.04.010
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
The regiospecific and enantioselective syntheses of various methylated regioisomers of epicatechin gallate (EGC) and epigallocatechin gallate (EGCG) have been achieved. (c) 2006 Elsevier Ltd. All rights reserved.
引用
收藏
页码:5897 / 5904
页数:8
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