Clean heterocyclic synthesis in water: I2/KI catalyzed one-pot synthesis of quinazolin-4(3H)-ones

被引：60

作者：

Bakavoli, Mehdi ^{[1
]}

Shiri, Ali ^{[1
]}

Ebrahimpour, Zahra ^{[1
]}

Rahimizadeh, Mohammad ^{[1
]}

机构：

[1] Ferdowsi Univ Mashhad, Sch Sci, Dept Chem, Mashhad 917751436, Iran

来源：

CHINESE CHEMICAL LETTERS | 2008年 / 19卷 / 12期

关键词：

Iodine; Quinazolinone; Cyclocondensation;

D O I：

10.1016/j.cclet.2008.07.016

中图分类号：

O6 [化学];

学科分类号：

0703 [化学];

摘要：

Oxidative cyclocondensation of o-aminobenzamide with various aldehydes in water using I-2/KI as catalyst and oxidizing agent is carried out giving the corresponding quinazolin-4(3H)-ones 3a-n in good to excellent yields. (c) 2008 Mehdi Bakavoli. Published by Elsevier B.V. on behalf of Chinese Chemical Society. All rights reserved.

引用

页码：1403 / 1406

页数：4

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