Microwave-assisted rapid synthesis of the cytotoxic alkaloid luotonin A

被引：111

作者：

Yadav, JS ^{[1
]}

Reddy, BVS ^{[1
]}

机构：

[1] Indian Inst Chem Technol, Organ Chem Div 1, Hyderabad 500007, Andhra Pradesh, India

来源：

TETRAHEDRON LETTERS | 2002年 / 43卷 / 10期

关键词：

deoxyvasinone; antitumor; quinazolines; microwave irradiation;

D O I：

10.1016/S0040-4039(02)00135-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The total synthesis of the cytotoxic alkaloid luotonin A has been achieved for the first time in high yields by the cyclocondensation of 3-oxo-1H-pyrrolo[3,4-b]quinoline with isatoic anhydride in solvent-free conditions Under microwave irradiation. (C) 2002 Elsevier Science Ltd. All rights reserved.

引用

页码：1905 / 1907

页数：3

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