An efficient access to 4-alkylidene-5,6-dihydro-4H-pyrrolo[1,2-c][1,2,3]triazoles

被引：23

作者：

Chen, Wan-li

Su, Chen-liang

Huang, Xian

机构：

[1] Zhejiang Univ, Dept Chem, Hangzhou 310028, Peoples R China

[2] Chinese Acad Sci, Shanghai Inst Organ Chem, State Key Lab Organomet Chem, Shanghai 200232, Peoples R China

来源：

SYNLETT | 2006年 / 09期

关键词：

1,2,3-trizaole; alkylidenecyclopropanes (MCPs); 1,3-dipolar; cycloaddition; Heck reaction;

D O I：

10.1055/s-2006-939708

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

From alkylidenecyclopropanes (MCPs), 4-alkylidene-5,6-dihydro-4H-pyrrolo-[1,2-c][1,2,3]triazoles 6 were prepared in moderate yields through diiodogenation, Cu(I)-catalyzed 1,3-dipolar cycloaddition and subsequent intramolecular Heck reaction.

引用

页码：1446 / 1448

页数：3

共 43 条

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