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Targeting c-kit mutations in solid tumors:: Scientific rationale and novel therapeutic options
被引:134
作者
:
Demetri, GD
论文数:
0
引用数:
0
h-index:
0
机构:
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Adult Oncol, Boston, MA 02115 USA
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Adult Oncol, Boston, MA 02115 USA
Demetri, GD
[
1
]
机构
:
[1]
Harvard Univ, Sch Med, Dana Farber Canc Inst, Dept Adult Oncol, Boston, MA 02115 USA
来源
:
SEMINARS IN ONCOLOGY
|
2001年
/ 28卷
/ 05期
关键词
:
D O I
:
10.1053/sonc.2001.29181
中图分类号
:
R73 [肿瘤学];
学科分类号
:
100214 ;
摘要
:
引用
收藏
页码:19 / 26
页数:8
相关论文
共 41 条
[21]
Mutations in exon 11 of c-kit occur preferentially in malignant versus benign gastrointestinal stromal tumors and do not occur in leiomyomas or leiomyosarcomas
Lasota, J
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Lasota, J
Jasinski, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Jasinski, M
Sarlomo-Rikala, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Sarlomo-Rikala, M
论文数:
引用数:
h-index:
机构:
Miettinen, M
[J].
AMERICAN JOURNAL OF PATHOLOGY,
1999,
154
(01)
: 53
-
60
[22]
KIT extracellular and kinase domain mutations in gastrointestinal stromal tumors
Lux, ML
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Lux, ML
Rubin, BP
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Rubin, BP
Biase, TL
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Biase, TL
Chen, CJ
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Chen, CJ
Maclure, T
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Maclure, T
论文数:
引用数:
h-index:
机构:
Demetri, G
Xiao, S
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Xiao, S
Singer, S
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Singer, S
Fletcher, CDM
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Fletcher, CDM
Fletcher, JA
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Fletcher, JA
[J].
AMERICAN JOURNAL OF PATHOLOGY,
2000,
156
(03)
: 791
-
795
[23]
Immunohistochemical spectrum of GISTs at different sites and their differential diagnosis with a reference to CD117 (KIT)
Miettinen, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Miettinen, M
Sobin, LH
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Sobin, LH
Sarlomo-Rikala, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Sarlomo-Rikala, M
[J].
MODERN PATHOLOGY,
2000,
13
(10)
: 1134
-
1142
[24]
Gastrointestinal stromal tumors: Recent advances in understanding of their biology
论文数:
引用数:
h-index:
机构:
Miettinen, M
Sarlomo-Rikala, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Sarlomo-Rikala, M
Lasota, J
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Lasota, J
[J].
HUMAN PATHOLOGY,
1999,
30
(10)
: 1213
-
1220
[25]
Gastrointestinal stromal tumors - definition, clinical, histological, immunohistochemical, and molecular genetic features and differential diagnosis
论文数:
引用数:
h-index:
机构:
Miettinen, M
Lasota, J
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Lasota, J
[J].
VIRCHOWS ARCHIV,
2001,
438
(01)
: 1
-
12
[26]
Familial gastrointestinal stromal tumours with germline mutation of the KIT gene
Nishida, T
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Nishida, T
Hirota, S
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Hirota, S
Taniguchi, M
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Taniguchi, M
Hashimoto, K
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Hashimoto, K
Isozaki, K
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Isozaki, K
Nakamura, H
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Nakamura, H
Kanakura, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Kanakura, Y
Tanaka, T
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Tanaka, T
Takabayashi, A
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Takabayashi, A
论文数:
引用数:
h-index:
机构:
Matsuda, H
Kitamura, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Kitamura, Y
[J].
NATURE GENETICS,
1998,
19
(04)
: 323
-
324
[27]
Nishida T, 2000, HISTOL HISTOPATHOL, V15, P1293, DOI 10.14670/HH-15.1293
[28]
Soft tissue leiomyosarcomas and malignant gastrointestinal stromal tumors: Differences in clinical outcome and expression of multidrug resistance proteins
Plaat, BEC
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Plaat, BEC
Hollema, H
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Hollema, H
Molenaar, WM
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Molenaar, WM
Broers, GHT
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Broers, GHT
Piipe, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Piipe, J
Mastik, MF
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Mastik, MF
Hoekstra, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Hoekstra, HJ
van den Berg, E
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
van den Berg, E
Scheper, RJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Scheper, RJ
van der Graaf, WTA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
van der Graaf, WTA
[J].
JOURNAL OF CLINICAL ONCOLOGY,
2000,
18
(18)
: 3211
-
3220
[29]
PRIMARY STRUCTURE OF C-KIT - RELATIONSHIP WITH THE CSF-1/PDGF RECEPTOR KINASE FAMILY ONCOGENIC ACTIVATION OF V-KIT INVOLVES DELETION OF EXTRACELLULAR DOMAIN AND C-TERMINUS
QIU, F
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CYTOGENET LAB,NEW YORK,NY 10021
QIU, F
RAY, P
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CYTOGENET LAB,NEW YORK,NY 10021
RAY, P
BROWN, K
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CYTOGENET LAB,NEW YORK,NY 10021
BROWN, K
BARKER, PE
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CYTOGENET LAB,NEW YORK,NY 10021
BARKER, PE
JHANWAR, S
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CYTOGENET LAB,NEW YORK,NY 10021
JHANWAR, S
RUDDLE, FH
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CYTOGENET LAB,NEW YORK,NY 10021
RUDDLE, FH
BESMER, P
论文数:
0
引用数:
0
h-index:
0
机构:
MEM SLOAN KETTERING CANC CTR,CYTOGENET LAB,NEW YORK,NY 10021
BESMER, P
[J].
EMBO JOURNAL,
1988,
7
(04)
: 1003
-
1011
[30]
Molecular insights into the histogenesis and pathogenesis of gastrointestinal stromal tumors
Rubin, BP
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Rubin, BP
Fletcher, JA
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Fletcher, JA
Fletcher, CDM
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Fletcher, CDM
[J].
INTERNATIONAL JOURNAL OF SURGICAL PATHOLOGY,
2000,
8
(01)
: 5
-
10
←
1
2
3
4
5
→
共 41 条
[21]
Mutations in exon 11 of c-kit occur preferentially in malignant versus benign gastrointestinal stromal tumors and do not occur in leiomyomas or leiomyosarcomas
Lasota, J
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Lasota, J
Jasinski, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Jasinski, M
Sarlomo-Rikala, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Sarlomo-Rikala, M
论文数:
引用数:
h-index:
机构:
Miettinen, M
[J].
AMERICAN JOURNAL OF PATHOLOGY,
1999,
154
(01)
: 53
-
60
[22]
KIT extracellular and kinase domain mutations in gastrointestinal stromal tumors
Lux, ML
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Lux, ML
Rubin, BP
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Rubin, BP
Biase, TL
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Biase, TL
Chen, CJ
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Chen, CJ
Maclure, T
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Maclure, T
论文数:
引用数:
h-index:
机构:
Demetri, G
Xiao, S
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Xiao, S
Singer, S
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Singer, S
Fletcher, CDM
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Fletcher, CDM
Fletcher, JA
论文数:
0
引用数:
0
h-index:
0
机构:
Brigham & Womens Hosp, Dept Pathol, Boston, MA 02115 USA
Fletcher, JA
[J].
AMERICAN JOURNAL OF PATHOLOGY,
2000,
156
(03)
: 791
-
795
[23]
Immunohistochemical spectrum of GISTs at different sites and their differential diagnosis with a reference to CD117 (KIT)
Miettinen, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Miettinen, M
Sobin, LH
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Sobin, LH
Sarlomo-Rikala, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Sarlomo-Rikala, M
[J].
MODERN PATHOLOGY,
2000,
13
(10)
: 1134
-
1142
[24]
Gastrointestinal stromal tumors: Recent advances in understanding of their biology
论文数:
引用数:
h-index:
机构:
Miettinen, M
Sarlomo-Rikala, M
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Sarlomo-Rikala, M
Lasota, J
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Lasota, J
[J].
HUMAN PATHOLOGY,
1999,
30
(10)
: 1213
-
1220
[25]
Gastrointestinal stromal tumors - definition, clinical, histological, immunohistochemical, and molecular genetic features and differential diagnosis
论文数:
引用数:
h-index:
机构:
Miettinen, M
Lasota, J
论文数:
0
引用数:
0
h-index:
0
机构:
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Armed Forces Inst Pathol, Dept Soft Tissue Pathol, Washington, DC 20306 USA
Lasota, J
[J].
VIRCHOWS ARCHIV,
2001,
438
(01)
: 1
-
12
[26]
Familial gastrointestinal stromal tumours with germline mutation of the KIT gene
Nishida, T
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Nishida, T
Hirota, S
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Hirota, S
Taniguchi, M
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Taniguchi, M
Hashimoto, K
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Hashimoto, K
Isozaki, K
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Isozaki, K
Nakamura, H
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Nakamura, H
Kanakura, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Kanakura, Y
Tanaka, T
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Tanaka, T
Takabayashi, A
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Takabayashi, A
论文数:
引用数:
h-index:
机构:
Matsuda, H
Kitamura, Y
论文数:
0
引用数:
0
h-index:
0
机构:
Osaka Univ, Sch Med, Dept Surg 1, Suita, Osaka 565, Japan
Kitamura, Y
[J].
NATURE GENETICS,
1998,
19
(04)
: 323
-
324
[27]
Nishida T, 2000, HISTOL HISTOPATHOL, V15, P1293, DOI 10.14670/HH-15.1293
[28]
Soft tissue leiomyosarcomas and malignant gastrointestinal stromal tumors: Differences in clinical outcome and expression of multidrug resistance proteins
Plaat, BEC
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Plaat, BEC
Hollema, H
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Hollema, H
Molenaar, WM
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Molenaar, WM
Broers, GHT
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Broers, GHT
Piipe, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Piipe, J
Mastik, MF
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Mastik, MF
Hoekstra, HJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Hoekstra, HJ
van den Berg, E
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
van den Berg, E
Scheper, RJ
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
Scheper, RJ
van der Graaf, WTA
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Groningen Hosp, Dept Pathol, NL-9700 RB Groningen, Netherlands
van der Graaf, WTA
[J].
JOURNAL OF CLINICAL ONCOLOGY,
2000,
18
(18)
: 3211
-
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