A synthesis of the derivatives of 1,2,3,5,10,10a-hexahydrobenz[f]indolizine-6,9-dione having antifungal activity as a simple model of saframycin A

被引：17

作者：

Kubo, A ^{[1
]}

Nakai, T ^{[1
]}

Koizumi, Y ^{[1
]}

Kitahara, Y ^{[1
]}

Saito, N ^{[1
]}

Mikami, Y ^{[1
]}

Yazawa, K ^{[1
]}

Uno, J ^{[1
]}

机构：

[1] CHIBA UNIV,RES CTR PATHOGEN FUNGI & MICROBIAL TOXICOSES,DIV EXPTL CHEMOTHERAPY,CHUO KU,CHIBA 280,JAPAN

来源：

HETEROCYCLES | 1996年 / 42卷 / 01期

关键词：

D O I：

10.3987/COM-94-S5-1

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A simple and efficient synthesis of 1,2,3,5,10,10a-hexahydrobenz[f]indolizine-6,9-dione (7) and its analogs (28-30) is described starting from the corresponding lactam (15b).

引用

页码：195 / 211

页数：17

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