An efficient, one-pot, synthesis of dithiocarbamates from the corresponding alcohols using Mitsunobu's reagent

被引：95

作者：

Chaturvedi, D

Ray, S

机构：

[1] Medicinal and Process Chemistry Division, Central Drug Research Institute

来源：

TETRAHEDRON LETTERS | 2006年 / 47卷 / 08期

关键词：

Mitsunobu's reagent; carbon disulfide; alcohols; dithiocarbamates; thiocarbamation;

D O I：

10.1016/j.tetlet.2005.12.079

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A Mitsunobu-based protocol has been developed for the synthesis of dithiocarbamates from the corresponding alcohols using carbon disulfide and amines in good to excellent yields. This protocol is mild, chemoselective and efficient compared to other reported methods. (c) 2005 Elsevier Ltd. All rights reserved.

引用

页码：1307 / 1309

页数：3

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