An expeditious approach to tri-substituted chiral thiazolines

被引：17

作者：

Abdel-Jalil, RJ ^{[1
]}

Saeed, M ^{[1
]}

Voelter, W ^{[1
]}

机构：

[1] Univ Tubingen, Inst Phys Chem, Phys Biochem Abt, D-72076 Tubingen, Germany

来源：

TETRAHEDRON LETTERS | 2001年 / 42卷 / 13期

关键词：

D O I：

10.1016/S0040-4039(01)00188-5

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A regio- and stereoselective route from the cis-oriented epoxytriflate pentoses 1 and 4 via 4-amino-4-deoxy sugars 2 and 5 to chiral thiazoline derivatives 3a-e and 6a-e in high yields is described. (C) 2001 Elsevier Science Ltd. All rights reserved.

引用

页码：2435 / 2437

页数：3

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