共 39 条
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N-arylaminonitriles as bioavailable peptidomimetic inhibitors of cathepsin B
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Greenspan, PD
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Clark, KL
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Cowen, SD
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McQuire, LW
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Tommasi, RA
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Farley, DL
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Quadros, E
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Coppa, DE
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Du, ZM
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Fang, Z
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Zhou, HH
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Doughty, J
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Toscano, KT
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Wigg, AM
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Zhou, SY
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BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2003, 13 (22)
:4121-4124

Greenspan, PD
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Clark, KL
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Cowen, SD
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

McQuire, LW
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Tommasi, RA
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Farley, DL
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Quadros, E
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Coppa, DE
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h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Du, ZM
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Fang, Z
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Zhou, HH
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Doughty, J
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Toscano, KT
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Wigg, AM
论文数: 0 引用数: 0
h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA

Zhou, SY
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h-index: 0
机构:
Novartis Inst Biomed Res, E Hanover, NJ 07936 USA Novartis Inst Biomed Res, E Hanover, NJ 07936 USA
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Identification of dipeptidyl nitriles as potent and selective inhibitors of cathepsin B through structure-based drug design
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Greenspan, PD
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Clark, KL
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Cowen, SD
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McQuire, LW
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Farley, DL
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van Duzer, JH
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Goldberg, RL
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Zhou, HH
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Du, ZM
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Fitt, JJ
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Coppa, DE
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Fang, Z
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Macchia, W
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Zhu, LJ
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Capparelli, MP
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Goldstein, R
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Wigg, AM
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JOURNAL OF MEDICINAL CHEMISTRY,
2001, 44 (26)
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Greenspan, PD
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Clark, KL
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Tommasi, RA
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Cowen, SD
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

McQuire, LW
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Farley, DL
论文数: 0 引用数: 0
h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

van Duzer, JH
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Goldberg, RL
论文数: 0 引用数: 0
h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Zhou, HH
论文数: 0 引用数: 0
h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Du, ZM
论文数: 0 引用数: 0
h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Fitt, JJ
论文数: 0 引用数: 0
h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Coppa, DE
论文数: 0 引用数: 0
h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Fang, Z
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Macchia, W
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Zhu, LJ
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Capparelli, MP
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Goldstein, R
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Wigg, AM
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Doughty, JR
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Bohacek, RS
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h-index: 0
机构:
Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA

Knap, AK
论文数: 0 引用数: 0
h-index: 0
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Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA Nova Pharmaceut Corp, Arthrit & Bone Metab Res, Summit, NJ 07901 USA
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Navia, MM
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Tanner, M
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Alonso, PL
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HANZLIK, RP
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ZYGMUNT, J
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机构: Department of Medicinal Chemistry, University of Kansas, Lawrence, KS

MOON, JB
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Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Lee, Ji H.
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Pandey, Kailash C.
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Univ Calif San Francisco, San Francisco Gen Hosp, Dept Med, San Francisco, CA 94143 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Harrison, Amanda
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Univ Calif San Francisco, San Francisco Gen Hosp, Dept Med, San Francisco, CA 94143 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Sajid, Mohammed
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Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA
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Shelat, Anang A.
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St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA

Obrien, Terri
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Univ Calif San Francisco, Dept Cellular & Mol Pharmacol, San Francisco, CA 94143 USA Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA

Caffrey, Conor R.
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Univ Calif San Francisco, Dept Cellular & Mol Pharmacol, San Francisco, CA 94143 USA Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA

Kosinski, Aaron
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h-index: 0
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St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA

Connelly, Michele
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St Jude Childrens Res Hosp, Dept Chem Biol & Therapeut, Memphis, TN 38105 USA Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA

Harbut, Michael
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Univ Penn, Dept Pharmacol, Philadelphia, PA 19146 USA Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA

Greenbaum, Doron
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Univ Penn, Dept Pharmacol, Philadelphia, PA 19146 USA Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA

McKerrow, James H.
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h-index: 0
机构:
Univ Calif San Francisco, Dept Cellular & Mol Pharmacol, San Francisco, CA 94143 USA Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA

Guy, R. Kiplin
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h-index: 0
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Univ Calif San Francisco, Grad Program Chem & Chem Biol, San Francisco, CA 94143 USA
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Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3LI, Canada Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3LI, Canada

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Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3LI, Canada Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3LI, Canada

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Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3LI, Canada Merck Frosst Ctr Therapeut Res, Dept Med Chem, Kirkland, PQ H9H 3LI, Canada

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Bryant, C
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机构: Celera Genom Inc, San Francisco, CA 94080 USA

Davis, DE
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机构: Celera Genom Inc, San Francisco, CA 94080 USA

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机构: Celera Genom Inc, San Francisco, CA 94080 USA

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机构: Celera Genom Inc, San Francisco, CA 94080 USA

Venkatraman, S
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h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA

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机构: Celera Genom Inc, San Francisco, CA 94080 USA

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机构: Celera Genom Inc, San Francisco, CA 94080 USA

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机构: Celera Genom Inc, San Francisco, CA 94080 USA

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Janc, JW
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机构: Celera Genom Inc, San Francisco, CA 94080 USA

Yu, ZW
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机构: Celera Genom Inc, San Francisco, CA 94080 USA

Percival, MD
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Prasit, P
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Oballa, R
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h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA

Riendeau, D
论文数: 0 引用数: 0
h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA

Young, RN
论文数: 0 引用数: 0
h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA

Wesolowski, G
论文数: 0 引用数: 0
h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA

Rodan, SB
论文数: 0 引用数: 0
h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA

Johnson, C
论文数: 0 引用数: 0
h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA

Kimmel, DB
论文数: 0 引用数: 0
h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA

Rodan, G
论文数: 0 引用数: 0
h-index: 0
机构: Celera Genom Inc, San Francisco, CA 94080 USA
[20]
A novel class of nonpeptidic biaryl inhibitors of human cathepsin K
[J].
Robichaud, J
;
Oballa, R
;
Prasit, P
;
Falgueyret, JP
;
Percival, MD
;
Wesolowski, G
;
Rodan, SB
;
Kimmel, D
;
Johnson, C
;
Bryant, C
;
Venkatraman, S
;
Setti, E
;
Mendonca, R
;
Palmer, JT
.
JOURNAL OF MEDICINAL CHEMISTRY,
2003, 46 (17)
:3709-3727

Robichaud, J
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Oballa, R
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Prasit, P
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Falgueyret, JP
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Percival, MD
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Wesolowski, G
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Rodan, SB
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Kimmel, D
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Johnson, C
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Bryant, C
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Venkatraman, S
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Setti, E
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Mendonca, R
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada

Palmer, JT
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Dept Chem, Quebec City, PQ H9H 3L1, Canada