The human CYP3A subfamily: Practical considerations

被引:183
作者
Wrighton, SA
Schuetz, EG
Thummel, KE
Shen, DD
Korzekwa, KR
Watkins, PB
机构
[1] Lilly Corp Ctr, Lilly Res Labs, Dept Drug Disposit, Indianapolis, IN 46285 USA
[2] St Jude Childrens Res Hosp, Dept Pharmaceut Sci, Memphis, TN 38105 USA
[3] Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA
[4] Univ Washington, Dept Pharm, Seattle, WA 98195 USA
[5] Camitro Corp, Menlo Pk, CA 94025 USA
[6] Univ N Carolina, Chapel Hill, NC 27599 USA
关键词
D O I
10.1081/DMR-100102338
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:339 / 361
页数:23
相关论文
共 104 条
[1]   DOSE OF MIDAZOLAM SHOULD BE REDUCED DURING DILTIAZEM AND VERAPAMIL TREATMENTS [J].
BACKMAN, JT ;
OLKKOLA, KT ;
ARANKO, K ;
HIMBERG, JJ ;
NEUVONEN, PJ .
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY, 1994, 37 (03) :221-225
[2]   Population distribution and effects on drug metabolism of a genetic variant in the 5′ promotor region of CYP3A4 [J].
Ball, SE ;
Scatina, JA ;
Kao, J ;
Ferron, GM ;
Fruncillo, R ;
Mayer, P ;
Weinryb, I ;
Guida, M ;
Hopkins, PJ ;
Warner, N ;
Hall, J .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1999, 66 (03) :288-294
[3]   Steroid transport, accumulation, and antagonism of P-glycoprotein in multidrug-resistant cells [J].
Barnes, KM ;
Dickstein, B ;
Cutler, GB ;
Fojo, T ;
Bates, SE .
BIOCHEMISTRY, 1996, 35 (15) :4820-4827
[4]   INHIBITION OF ALFENTANIL METABOLISM BY ERYTHROMYCIN [J].
BARTKOWSKI, RR ;
GOLDBERG, ME ;
LARIJANI, GE ;
BOERNER, T .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1989, 46 (01) :99-102
[5]   ISOLATION AND SEQUENCE DETERMINATION OF A CDNA CLONE RELATED TO HUMAN CYTOCHROME-P-450 NIFEDIPINE OXIDASE [J].
BEAUNE, PH ;
UMBENHAUER, DR ;
BORK, RW ;
LLOYD, RS ;
GUENGERICH, FP .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1986, 83 (21) :8064-8068
[6]  
BENET LZ, 1996, GOODMAN GILMANS PHAR, P14
[7]   Assessment of the potential for a pharmacokinetic interaction between fluoxetine and terfenadine [J].
Bergstrom, RF ;
Goldberg, MJ ;
Cerimele, BJ ;
Hatcher, BL .
CLINICAL PHARMACOLOGY & THERAPEUTICS, 1997, 62 (06) :643-651
[8]   Identification of a human nuclear receptor defines a new signaling pathway for CYP3A induction [J].
Bertilsson, G ;
Heidrich, J ;
Svensson, K ;
Åsman, M ;
Jendeberg, L ;
Sydow-Bäckman, M ;
Ohlsson, R ;
Postlind, H ;
Blomquist, P ;
Berkenstam, A .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1998, 95 (21) :12208-12213
[9]   SXR, a novel steroid and xenobiotic-sensing nuclear receptor [J].
Blumberg, B ;
Sabbagh, W ;
Juguilon, H ;
Bolado, J ;
van Meter, CM ;
Ono, ES ;
Evans, RM .
GENES & DEVELOPMENT, 1998, 12 (20) :3195-3205
[10]  
BROWN MB, 1997, J CLIN INVEST, V99, P2545