A general synthesis of beta-aryl and heteroarylpyrroles by palladium-catalyzed coupling reaction of beta-tributylstannylpyrrole with aryl and heteroaryl halides

被引：20

作者：

Wang, JJ ^{[1
]}

Scott, AI ^{[1
]}

机构：

[1] TEXAS A&M UNIV,DEPT CHEM,CTR BIOL NMR,COLLEGE STN,TX 77843

来源：

TETRAHEDRON LETTERS | 1996年 / 37卷 / 19期

关键词：

D O I：

10.1016/0040-4039(96)00530-8

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Several beta-aryl and heteroarylpyrroles have been synthesized by palladium-catalyzed coupling reaction of beta-tributylstannylpyrroles with aryl and heteroaryl halides in 62-89% yields. These precursors may be readily converted into beta-aryl and heteroaryl substituted porphyrins for the study of the oxophlorin to oxaporphyrin conversion in heme catabolism, catalyzed by heme oxygenase. (C) 1996 Elsevier Science Ltd.

引用

页码：3247 / 3250

页数：4

共 6 条

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[6] AN EFFICIENT SYNTHESIS OF 3-VINYLPYRROLES BY STILLE COUPLING REACTION OF 3-IODOPYRROLES WITH VINYLTRIBUTYLTIN
WANG, JJ
SCOTT, AI
[J]. TETRAHEDRON LETTERS, 1995, 36 (39) : 7043 - 7046

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