Iodination of aromatic residues in peptides by reaction with IPy(2)BF(4)

被引：39

作者：

Barluenga, J ^{[1
]}

GarciaMartin, MA ^{[1
]}

Gonzalez, JM ^{[1
]}

Clapes, P ^{[1
]}

Valencia, G ^{[1
]}

机构：

[1] CSIC,UNIT PROT CHEM & BIOCHEM,CTR INVEST & DESARROLLO,E-08034 BARCELONA,SPAIN

来源：

CHEMICAL COMMUNICATIONS | 1996年 / 13期

关键词：

D O I：

10.1039/cc9960001505

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A simple and straightforward approach to selectively iodinate Tyr residues on peptides using IPy(2)BF(4) is described which is compatible with Met residues on the side chain; preliminary studies reveal that the method is also suitable to iodinate Phe derivatives.

引用

页码：1505 / 1506

页数：2

共 12 条

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