Pharmacotherapeutic potential of omega-conotoxin MVIIA (SNX-111), an N-type neuronal calcium channel blocker found in the venom of Conus magus

被引:90
作者
Bowersox, SS [1 ]
Luther, R [1 ]
机构
[1] Neurex Corp, Dept Pharmacol, Menlo Pk, CA 94025 USA
关键词
D O I
10.1016/S0041-0101(98)00158-5
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:1651 / 1658
页数:8
相关论文
共 32 条
[1]   SOLUTION STRUCTURE OF OMEGA-CONOTOXIN MVIIA USING 2D NMR-SPECTROSCOPY [J].
BASUS, VJ ;
NADASDI, L ;
RAMACHANDRAN, J ;
MILJANICH, GP .
FEBS LETTERS, 1995, 370 (03) :163-169
[2]  
Bowersox Scott, 1998, Drugs of the Future, V23, P152, DOI 10.1358/dof.1998.023.02.443399
[3]  
Bowersox SS, 1997, BRAIN RES, V747, P343
[4]  
Bowersox SS, 1996, J PHARMACOL EXP THER, V279, P1243
[5]   Use of intrathecal SNX-111, a novel, N-type, voltage-sensitive, calcium channel blocker, in the management of intractable brachial plexus avulsion pain [J].
Brose, WG ;
Gutlove, DP ;
Luther, RR ;
Bowersox, SS ;
McGuire, D .
CLINICAL JOURNAL OF PAIN, 1997, 13 (03) :256-259
[6]   A SELECTIVE N-TYPE CA2+-CHANNEL BLOCKER PREVENTS CA1 INJURY 24-H FOLLOWING SEVERE FOREBRAIN ISCHEMIA AND REDUCES INFARCTION FOLLOWING FOCAL ISCHEMIA [J].
BUCHAN, AM ;
GERTLER, SZ ;
LI, H ;
XUE, D ;
HUANG, ZG ;
CHAUNDY, KE ;
BARNES, K ;
LESIUK, HJ .
JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM, 1994, 14 (06) :903-910
[7]  
CHOI DW, 1995, TRENDS NEUROSCI, V18, P58
[8]  
CHUNG D, 1995, INT J PEPT PROT RES, V46, P320
[9]   SOLUTION STRUCTURE OF OMEGA-CONOTOXIN GVIA USING 2-D NMR-SPECTROSCOPY AND RELAXATION MATRIX ANALYSIS [J].
DAVIS, JH ;
BRADLEY, EK ;
MILJANICH, GP ;
NADASDI, L ;
RAMACHANDRAN, J ;
BASUS, VJ .
BIOCHEMISTRY, 1993, 32 (29) :7396-7405
[10]   SOLUTION STRUCTURE OF OMEGA-CONOTOXIN MVIIC, A HIGH-AFFINITY LIGAND OF P-TYPE CALCIUM CHANNELS, USING H-1-NMR SPECTROSCOPY AND COMPLETE RELAXATION MATRIX ANALYSIS [J].
FARRJONES, S ;
MILJANICH, GP ;
NADASDI, L ;
RAMACHANDRAN, J ;
BASUS, VJ .
JOURNAL OF MOLECULAR BIOLOGY, 1995, 248 (01) :106-124