A synthesis of the platelet aggregation inhibitor xemilofiban from L-aspartic acid. Confirmation of the absolute configuration.

被引:8
作者
Boys, ML [1 ]
机构
[1] GD Searle & Co, Dept Chem Sci, Skokie, IL 60077 USA
关键词
D O I
10.1016/S0040-4039(98)00602-9
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A synthesis of xemilofiban (SC-54684A) from L-aspartic acid has been achieved in an overall yield of 18 %, and the absolute configuration has been confirmed, (C) 1998 Elsevier Science Ltd. All rights reserved.
引用
收藏
页码:3449 / 3450
页数:2
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