Synthesis of indole-2-carboxylic acid esters

被引：4

作者：

Allen, DA ^{[1
]}

机构：

[1] Roche Biosci, Palo Alto, CA 94304 USA

来源：

SYNTHETIC COMMUNICATIONS | 1999年 / 29卷 / 03期

关键词：

D O I：

10.1080/00397919908085787

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The title compounds were prepared via lateral lithiation of N-Boc protected toluidines with sec-BuLi, quench with diethyl oxalate, followed by dehydration in TFA/CH2Cl2.

引用

页码：447 / 455

页数：9

共 16 条

[11] BENZAZEPINONE CALCIUM-CHANNEL BLOCKERS .4. STRUCTURE ACTIVITY OVERVIEW AND INTRACELLULAR BINDING-SITE
KIMBALL, SD
FLOYD, DM
DAS, J
HUNT, JT
KRAPCHO, J
ROVNYAK, G
DUFF, KJ
LEE, VG
MOQUIN, RV
TURK, CF
HEDBERG, SA
MORELAND, S
BRITTAIN, RJ
MCMULLEN, DM
NORMANDIN, DE
CUCINOTTA, GG
[J]. JOURNAL OF MEDICINAL CHEMISTRY, 1992, 35 (04) : 780 - 793
[12] ALPHA-KETO DIANIONS - NEW REACTIVE INTERMEDIATES
KOWALSKI, CJ
ODOWD, ML
BURKE, MC
FIELDS, KW
[J]. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 1980, 102 (16) : 5411 - 5412
[13] ORTHO FUNCTIONALIZATION OF N-(TERT-BUTOXYCARBONYL)ANILINE
MUCHOWSKI, JM
VENUTI, MC
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1980, 45 (23) : 4798 - 4801
[14] IRON-AMMONIUM CHLORIDE - A CONVENIENT AND INEXPENSIVE REDUCTANT
RAMADAS, K
SRINIVASAN, N
[J]. SYNTHETIC COMMUNICATIONS, 1992, 22 (22) : 3189 - 3195
[15] GENERATION AND REACTIONS OF 3-LITHIO-1-(PHENYLSULFONYL)INDOLE
SAULNIER, MG
GRIBBLE, GW
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1982, 47 (05) : 757 - 761
[16] SYNTHESES WITH N-PROTECTED 2-LITHIOINDOLES
SUNDBERG, RJ
RUSSELL, HF
[J]. JOURNAL OF ORGANIC CHEMISTRY, 1973, 38 (19) : 3324 - 3330

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