Comparative QSAR analysis of estrogen receptor ligands

被引：266

作者：

Gao, H

Katzenellenbogen, JA

Garg, R

Hansch, C ^{[1
]}

机构：

[1] Pomona Coll, Dept Chem, Claremont, CA 91711 USA

[2] Univ Illinois, Dept Chem, Urbana, IL 61801 USA

来源：

CHEMICAL REVIEWS | 1999年 / 99卷 / 03期

关键词：

D O I：

10.1021/cr980018g

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

[No abstract available]

引用

页码：723 / 744

页数：22

共 86 条

[1] THE USE OF CHARACTERISTIC VOLUMES TO MEASURE CAVITY TERMS IN REVERSED PHASE LIQUID-CHROMATOGRAPHY [J].

ABRAHAM, MH ;

MCGOWAN, JC .

CHROMATOGRAPHIA, 1987, 23 (04) :243-246

[2]

*AM CHEM SOC FACTS, 1998, CANC STAT

[3] OPTIMIZING OF 2,3-DIARYLINDENES AS FLUORESCENT ESTROGENS - VARIATION OF THE ACCEPTOR GROUP, ORTHO SUBSTITUTION OF THE 2-RING, AND C-1 METHYLATION [J].

ANSTEAD, GM ;

KATZENELLENBOGEN, JA .

JOURNAL OF MEDICINAL CHEMISTRY, 1988, 31 (09) :1754-1761

[4] 2-ARYLINDENES AND 2-ARYLINDENONES - MOLECULAR-STRUCTURES AND CONSIDERATIONS IN THE BINDING ORIENTATION OF UNSYMMETRICAL NONSTEROIDAL LIGANDS TO THE ESTROGEN-RECEPTOR [J].

ANSTEAD, GM ;

WILSON, SR ;

KATZENELLENBOGEN, JA .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (09) :2163-2171

[5] The estradiol pharmacophore: Ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site [J].

Anstead, GM ;

Carlson, KE ;

Katzenellenbogen, JA .

STEROIDS, 1997, 62 (03) :268-303

[6] KINETICS OF THE HORMONE-RECEPTOR INTERACTION - COMPETITION EXPERIMENTS WITH SLOWLY EQUILIBRATING LIGANDS [J].

ARANYI, P .

BIOCHIMICA ET BIOPHYSICA ACTA, 1980, 628 (02) :220-227

[7]

BARNETT V, 1984, STAT DATA

[8] REGIO AND STEREOSPECIFIC SYNTHESIS OF 11-BETA-SUBSTITUTED 19-NORSTEROIDS - INFLUENCE OF 11-BETA-SUBSTITUTION ON PROGESTERONE-RECEPTOR AFFINITY [J].

BELANGER, A ;

PHILIBERT, D ;

TEUTSCH, G .

STEROIDS, 1981, 37 (04) :361-382

[9] EFFECT OF TRIPHENYLACRYLONITRILE DERIVATIVES ON ESTRADIOL-RECEPTOR BINDING AND ON HUMAN-BREAST CANCER CELL-GROWTH [J].

BIGNON, E ;

PONS, M ;

DEPAULET, AC ;

DORE, JC ;

GILBERT, J ;

ABECASSIS, J ;

MIQUEL, JF ;

OJASOO, T ;

RAYNAUD, JP .

JOURNAL OF MEDICINAL CHEMISTRY, 1989, 32 (09) :2092-2103

[10] CRYSTAL-STRUCTURE OF THE LIGAND-BINDING DOMAIN OF THE HUMAN NUCLEAR RECEPTOR RXR-ALPHA [J].

BOURGUET, W ;

RUFF, M ;

CHAMBON, P ;

GRONEMEYER, H ;

MORAS, D .

NATURE, 1995, 375 (6530) :377-382

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